SCHEMBL5301989

SCHEMBL5301989

O=[N+]([O-])c1ccc(Cl)nc1NCc1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.55
CTSB P07858 1/20 0.55
PKM P14618 2/20 0.51
TXNRD1 Q16881 2/20 0.49
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
JAK2 O60674 1/20 0.42
IGF1R P08069 1/20 0.42
PIM1 P11309 1/20 0.42
SRC P12931 1/20 0.42
CSNK2A2 P19784 1/20 0.42
KCNA5 P22460 1/20 0.42
JAK1 P23458 1/20 0.42
CCNE1 P24864 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1917607 0.84 PIN1 (0.57) CTSBPKMKDM4EALDH1A1HPGD
SCHEMBL8134885 0.82 PKM (0.61) MAPTCTSBPKMKDM4EALDH1A1
SCHEMBL9537830 0.81 TXNRD1 (0.52) MAPTCTSBPKMTXNRD1ALDH1A1
SCHEMBL18319382 0.81 MAPT (0.64) MAPTTXNRD1KDM4EALDH1A1HPGD
SCHEMBL5301730 0.79 CTSB (0.49) MAPTCTSBPKMMAOAMAOB
SCHEMBL4892092 0.79 MAPT (0.55) MAPTTXNRD1KDM4EALDH1A1HTT
SCHEMBL2272150 0.79 MAPT (0.60) MAPTPKMTXNRD1KDM4EALDH1A1
SCHEMBL3332328 0.77 HPGD (0.49) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL6870152 0.77 CTSB (0.49) MAPTCTSBPKMKDM4EALDH1A1
SCHEMBL1330877 0.76 MAPT (0.49) MAPTPKMALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007020521-A1 PYRIDOYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2007-02-22 WO disclosed
US-5066654-A 2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants A. H. ROBINS COMPANY, INCORPORATED (US) 1991-11-19 US disclosed