SCHEMBL5305019

SCHEMBL5305019

O=[N+]([O-])c1cc(Cl)c(Cl)cc1Cn1cncn1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.45
CCR2 P41597 1/20 0.45
CCR4 P51679 1/20 0.45
PKM P14618 1/20 0.43
CYP19A1 P11511 9/20 0.41
STS P08842 2/20 0.39
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450404 0.83 CCR1 (0.51) CCR1CCR2CCR4PKMCYP19A1
SCHEMBL9525426 0.78 KDM4E (0.50) PKMCYP19A1STSALDH1A1HDAC1
SCHEMBL31005997 0.78 PKM (0.44) CCR1CCR2CCR4PKMCYP19A1
SCHEMBL14610826 0.76 CCR1 (0.40) CCR1CCR2CCR4MEN1ALDH1A1
SCHEMBL14610754 0.74 CYP19A1 (0.46) CCR1CCR2CCR4PKMCYP19A1
SCHEMBL994055 0.70 CYP19A1 (0.57) PKMCYP19A1MEN1KMT2AHDAC1
SCHEMBL6280404 0.69 PKM (0.49) PKMCYP19A1ALDH1A1HDAC1HDAC6
SCHEMBL11127500 0.69 PDK1 (0.46) ALDH1A1
SCHEMBL18138458 0.69 TSHR (0.44) ALDH1A1
SCHEMBL9747728 0.68 CCR1 (0.55) CCR1CCR2CCR4PKMCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007014054-A2 BENZENESULFONAMIDE INHIBITOR OF CCR2 CHEMOKINE RECEPTOR GLAXO GROUP LIMTED (GB) 2007-02-01 WO disclosed
WO-2007014054-A2 BENZENESULFONAMIDE INHIBITOR OF CCR2 CHEMOKINE RECEPTOR GLAXO GROUP LIMTED (GB) 2007-02-01 WO disclosed