SCHEMBL5315965

SCHEMBL5315965

CC(=O)NCc1c(F)cc(C#N)cc1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SETDB1 Q15047 1/20 0.43
ENPP2 Q13822 1/20 0.41
EGLN2 Q96KS0 2/20 0.38
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 1/20 0.34
GPR35 Q9HC97 1/20 0.34
EPHX2 P34913 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
STING1 Q86WV6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18300420 0.85 GPR35 (0.39) ENPP2ALDH1A1KMT2AGPR35EPHX2
SCHEMBL5315960 0.83 ENPP2 (0.39) ENPP2ALDH1A1KMT2AGPR35EPHX2
SCHEMBL25840301 0.80 ALDH1A1 (0.50) ALDH1A1NPSR1KMT2AEPHX2CYP1A2
SCHEMBL5318967 0.80 SETDB1 (0.55) SETDB1ENPP2EGLN2EPHX2
SCHEMBL18300223 0.79 CTSS (0.41) ENPP2EGLN2LMNA
SCHEMBL10622670 0.74 EGLN2 (0.41) EGLN2ALDH1A1KMT2AGPR35
SCHEMBL14232838 0.73 NPSR1 (0.53) NPSR1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL17514852 0.73 TTR (0.38) ALDH1A1KMT2ALMNA
SCHEMBL12845232 0.71 TTR (0.39) ALDH1A1KMT2AGPR35CYP3A4
SCHEMBL5315293 0.70 LOXL2 (0.60) SETDB1EGLN2ALDH1A1KMT2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3280707-B1 BICYCLIC QUINAZOLINONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2023-12-20 EP claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO disclosed