SCHEMBL5325359

SCHEMBL5325359

Cc1c(N)ccc(OCC(O)C(C)(C)O)c1F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
HSD17B10 Q99714 3/20 0.41
GLA P06280 2/20 0.41
GAA P10253 2/20 0.41
POLB P06746 1/20 0.38
CYP3A4 P08684 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 2/20 0.37
MAPK1 P28482 1/20 0.37
BLM P54132 1/20 0.37
TSHR P16473 1/20 0.37
AR P10275 9/20 0.34
VDR P11473 6/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323891 1.00 KDM4E (0.41) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL5326367 0.79 VDR (0.37) KDM4EALDH1A1HSD17B10VDR
SCHEMBL5323899 0.79 AAK1 (0.37) VDR
SCHEMBL5325348 0.78 L3MBTL1 (0.43) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL5323314 0.74 KMT2A (0.44) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL5327068 0.74 KMT2A (0.44) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL34472182 0.73 KDM4E (0.33) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL634310 0.67 ALDH1A1 (0.47) KDM4EALDH1A1HSD17B10GAAPOLB
SCHEMBL17353507 0.66 ALDH1A1 (0.49) KDM4EALDH1A1HSD17B10GAAPOLB
SCHEMBL2872256 0.66 ALDH1A1 (0.45) KDM4EALDH1A1HSD17B10GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121416-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-25 WO disclosed
WO-2007121416-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-25 WO disclosed