SCHEMBL5326735

SCHEMBL5326735

COc1ccc(-c2[c]cccc2)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
IMPDH2 P12268 1/20 0.47
IMPDH1 P20839 1/20 0.47
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.47
AR P10275 6/20 0.46
PGR P06401 2/20 0.46
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
F11 P03951 1/20 0.41
CHEK1 O14757 1/20 0.39
PRKCQ Q04759 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5322067 0.81 PDE4A (0.50) ALDH1A1KDM4EUSP2
SCHEMBL5329094 0.78 KDM4E (0.40) KDM4E
SCHEMBL29123961 0.78 MAOB (0.57) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL5330919 0.77 CNR2 (0.44) ARPGR
SCHEMBL5326419 0.77 CYP11B2 (0.44) ALDH1A1AR
SCHEMBL5327982 0.77 CYP11B2 (0.50)
SCHEMBL5321545 0.77 PTGS2 (0.46) ALDH1A1KDM4E
SCHEMBL5326742 0.76 ALDH1A1 (0.54) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL5327699 0.73 AR (0.47) IMPDH2IMPDH1ARMAOAMAOB
SCHEMBL5326185 0.73 AR (0.43) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135527-A2 BENZIMIDAZOLYL COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-11-29 WO claimed
WO-2007135529-A2 AZABENZIMIDAZOLYL COMPOUNDS AS MGLUR2 POTENTIATORS PFIZER PRODUCTS INC. (US) 2007-11-29 WO claimed
WO-2007135527-A2 BENZIMIDAZOLYL COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-11-29 WO disclosed
WO-2007135529-A2 AZABENZIMIDAZOLYL COMPOUNDS AS MGLUR2 POTENTIATORS PFIZER PRODUCTS INC. (US) 2007-11-29 WO disclosed