SCHEMBL53274

SCHEMBL53274

Nc1cc(C(c2ccc(O)c(N)c2)(C(F)(F)F)C(F)(F)F)ccc1O.O=C1OC(=O)c2cc(Oc3ccc4c(c3)C(=O)OC4=O)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
RECQL P46063 2/20 0.36
KMT2A Q03164 2/20 0.36
PKM P14618 1/20 0.36
ATM Q13315 1/20 0.35
CHEK1 O14757 1/20 0.34
FYN P06241 1/20 0.34
PDGFRB P09619 1/20 0.34
PIM1 P11309 1/20 0.34
FGFR1 P11362 1/20 0.34
FLT1 P17948 1/20 0.34
GRK5 P34947 1/20 0.34
MAP2K2 P36507 1/20 0.34
MAPK8 P45983 1/20 0.34
CDK8 P49336 1/20 0.34
RPS6KA3 P51812 1/20 0.34
PRKX P51817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849209 0.86 MAOA (0.40) MAPTALDH1A1ATMMAOAMAOB
SCHEMBL16594065 0.86 NR1H4 (0.31) MAPTATML3MBTL1NPSR1
SCHEMBL2607322 0.83 MAOA (0.43) MAPTALDH1A1ATMMAOAMAOB
SCHEMBL1553198 0.78 ALDH1A1 (0.46) MAPTMEN1ALDH1A1GAARECQL
SCHEMBL30175421 0.78 ALDH1A1 (0.46) MAPTMEN1ALDH1A1GAARECQL
SCHEMBL15699449 0.77 SRD5A2 (0.41) MEN1KMT2AMAPK14MAOAMAOB
SCHEMBL49774 0.76 ALOX15 (0.43) MAPTALDH1A1ATMTDP1MCL1
SCHEMBL18180026 0.76 MAOA (0.37) MAPTALDH1A1ATMMAOAMAOB
SCHEMBL26579 0.76 ALDH1A1 (0.59) MAPTMEN1ALDH1A1GAARECQL
SCHEMBL29360962 0.76 ALDH1A1 (0.59) MAPTMEN1ALDH1A1GAARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8613362-B2 Polymer membranes derived from aromatic polyimide membranes UOP LLC (US) 2013-12-24 US claimed
US-8561812-B2 Blend polymer membranes comprising thermally rearranged polymers derived from aromatic polyimides containing ortho-positioned functional groups UOP LLC (US) 2013-10-22 US claimed
US-20120276300-A1 POLYMER MEMBRANES PREPARED FROM AROMATIC POLYIMIDE MEMBRANES BY THERMAL TREATING AND UV CROSSLINKING UOP LLC (US) 2012-11-01 US claimed
US-20120085233-A1 BLEND POLYMER MEMBRANES COMPRISING THERMALLY REARRANGED POLYMERS DERIVED FROM AROMATIC POLYIMIDES CONTAINING ORTHO-POSITIONED FUNCTIONAL GROUPS UOP LLC (US) 2012-04-12 US claimed
EP-2411131-A2 POLYMER MEMBRANES PREPARED FROM AROMATIC POLYIMIDE MEMBRANES BY THERMAL TREATING AND UV CROSSLINKING UOP LLC (US) 2012-02-01 EP claimed
EP-2411130-A2 HIGH PERFORMANCE CROSS-LINKED POLYBENZOXAZOLE AND POLYBENZOTHIAZOLE POLYMER MEMBRANES UOP LLC (US) 2012-02-01 EP claimed
EP-2411132-A2 POLYMER MEMBRANES DERIVED FROM AROMATIC POLYIMIDE MEMBRANES UOP LLC (US) 2012-02-01 EP claimed
EP-2411455-A2 BLEND POLYMER MEMBRANES COMPRISING THERMALLY REARRANGED POLYMERS DERIVED FROM AROMATIC POLYIMIDES CONTAINING ORTHO-POSITIONED FUNCTIONAL GROUPS UOP LLC (US) 2012-02-01 EP claimed
WO-2011163293-A2 PROCESS OF MAKING ASYMMETRIC POLYBENZOXAZOLE MEMBRANES UOP LLC (US) 2011-12-29 WO claimed
US-20110316181-A1 PROCESS OF MAKING ASYMMETRIC POLYBENZOXAZOLE MEMBRANES UOP LLC (US) 2011-12-29 US claimed
US-20100242723-A1 Blend Polymer Membranes Comprising Thermally Rearranged Polymers Derived from Aromatic Polyimides Containing Ortho-Positioned Functional Groups UOP LLC 2010-09-30 US claimed
WO-2010110975-A2 HIGH PERFORMANCE CROSS-LINKED POLYBENZOXAZOLE AND POLYBENZOTHIAZOLE POLYMER MEMBRANES UOP LLC (US) 2010-09-30 WO claimed
WO-2010110994-A2 POLYMER MEMBRANES PREPARED FROM AROMATIC POLYIMIDE MEMBRANES BY THERMAL TREATING AND UV CROSSLINKING UOP LLC (US) 2010-09-30 WO claimed
WO-2010110986-A2 POLYBENZOXAZOLE POLYMER-BASED MIXED MATRIX MEMBRANES UOP LLC (US) 2010-09-30 WO claimed
WO-2010110995-A2 POLYMER MEMBRANES DERIVED FROM AROMATIC POLYIMIDE MEMBRANES UOP LLC (US) 2010-09-30 WO claimed
US-20100243567-A1 Polymer Membranes Derived from Aromatic Polyimide Membranes UOP LLC 2010-09-30 US claimed
WO-2010110968-A2 BLEND POLYMER MEMBRANES COMPRISING THERMALLY REARRANGED POLYMERS DERIVED FROM AROMATIC POLYIMIDES CONTAINING ORTHO-POSITIONED FUNCTIONAL GROUPS UOP LLC (US) 2010-09-30 WO claimed
US-20100133190-A1 METHOD TO IMPROVE THE SELECTIVITY OF POLYBENZOXAZOLE MEMBRANES UOP LLC (US) 2010-06-03 US claimed
US-20100133192-A1 Polymer Membranes Prepared from Aromatic Polyimide Membranes by Thermal Treating and UV Crosslinking UOP LLC 2010-06-03 US claimed
US-20100137124-A1 High Performance Cross-Linked Polybenzoxazole and Polybenzothiazole Polymer Membranes UOP LLC 2010-06-03 US claimed