SCHEMBL533018

SCHEMBL533018

Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)c1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
MEN1 O00255 1/20 0.51
TSHR P16473 1/20 0.51
KMT2A Q03164 1/20 0.51
ATM Q13315 1/20 0.51
ERAP1 Q9NZ08 1/20 0.51
LMNA P02545 4/20 0.49
GLA P06280 1/20 0.49
MCL1 Q07820 8/20 0.47
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
TP53 P04637 2/20 0.43
POLB P06746 2/20 0.43
MAPT P10636 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
HTT P42858 1/20 0.40
CCKBR P32239 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533942 0.85 L3MBTL1 (0.48) ALDH1A1L3MBTL1MEN1TSHRKMT2A
SCHEMBL534052 0.82 MEN1 (0.47) ALDH1A1L3MBTL1MEN1TSHRKMT2A
SCHEMBL533043 0.82 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ALMNATP53
SCHEMBL532999 0.79 TP53 (0.48) ALDH1A1MEN1KMT2AHCRTR1TP53
SCHEMBL533091 0.78 BRPF1 (0.52) ALDH1A1MEN1KMT2ALMNATP53
SCHEMBL532951 0.78 EDNRB (0.45) ALDH1A1L3MBTL1MEN1KMT2ALMNA
SCHEMBL533247 0.76 CNR2 (0.39) KMT2AERAP1TP53POLBMAPT
SCHEMBL532980 0.76 JAK2 (0.48) ALDH1A1L3MBTL1MEN1TSHRKMT2A
SCHEMBL533656 0.76 ACLY (0.39) L3MBTL1KMT2ALMNAPOLBMAPT
SCHEMBL532038 0.75 ALDH1A1 (0.54) ALDH1A1TSHRKMT2ALMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed