SCHEMBL533043

SCHEMBL533043

COc1ccc(Cl)c(S(=O)(=O)Nc2c(C)cc(C)c(N3CCCC3)c2C)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
MAPT P10636 3/20 0.43
RECQL P46063 1/20 0.43
FFAR4 Q5NUL3 2/20 0.42
PKM P14618 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 3/20 0.41
HTT P42858 2/20 0.41
FBP1 P09467 1/20 0.40
TP53 P04637 2/20 0.40
SGK1 O00141 2/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532935 0.88 ALDH1A1 (0.53) ALDH1A1MAPTRECQLSMN1; SMN2LMNA
SCHEMBL533942 0.86 L3MBTL1 (0.48) ALDH1A1MAPTRECQLSMN1; SMN2LMNA
SCHEMBL534052 0.83 MEN1 (0.47) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL532953 0.83 FFAR4 (0.59) ALDH1A1MAPTFFAR4PKMSMN1; SMN2
SCHEMBL533018 0.82 ALDH1A1 (0.51) ALDH1A1MAPTSMN1; SMN2LMNAMEN1
SCHEMBL14288678 0.80 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL533676 0.80 ACLY (0.46) ALDH1A1MAPTFFAR4SMN1; SMN2LMNA
SCHEMBL532951 0.78 EDNRB (0.45) ALDH1A1MAPTFFAR4SMN1; SMN2LMNA
SCHEMBL534062 0.78 ERAP1 (0.52) ALDH1A1RECQLSMN1; SMN2LMNAMEN1
SCHEMBL532936 0.78 MCOLN3 (0.51) ALDH1A1PKMSMN1; SMN2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed