Omidenepag

Omidenepag

SCHEMBL533245

O=C(O)CNc1cccc(CN(Cc2ccc(-n3cccn3)cc2)S(=O)(=O)c2cccnc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGER2

The experimentally established mechanism targets of Omidenepag. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGER2 known ✓ P43116 20/20 1.00
PTGER4 P35408 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Omidenepag SCHEMBL30433956 1.00 PTGER2 (1.00) PTGER2PTGER4
Omidenepag SCHEMBL29565501 1.00 PTGER2 (1.00) PTGER2PTGER4
Omidenepag SCHEMBL533632 1.00 PTGER2 (1.00) PTGER2PTGER4
SCHEMBL22364205 0.89 PTGER2 (0.81) PTGER2PTGER4
SCHEMBL534263 0.89 PTGER2 (1.00) PTGER2PTGER4
Omidenepag Isopropyl SCHEMBL30434740 0.89 PTGER2 (1.00) PTGER2PTGER4
Omidenepag Isopropyl SCHEMBL15414827 0.89 PTGER2 (1.00) PTGER2PTGER4
Omidenepag Isopropyl SCHEMBL29375346 0.89 PTGER2 (1.00) PTGER2PTGER4
SCHEMBL22283788 0.88 PTGER2 (0.79) PTGER2PTGER4
SCHEMBL533704 0.88 PTGER2 (0.79) PTGER2PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 124 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11974994-B2 Agent for treating or preventing glaucoma including a sulfonamide compound and another drug SANTEN PHARMACEUTICAL CO., LTD. (JP) 2024-05-07 US claimed
US-20240024484-A1 PHARMACEUTICAL COMPOSITION CONTAINING PYRIDYLAMINOACETIC ACID COMPOUND SANTEN PHARMACEUTICAL CO., LTD. (JP) 2024-01-25 US claimed
US-20240000763-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A PYRIDYLAMINOACETIC ACID COMPOUND SANTEN PHARMACEUTICAL CO., LTD. (JP) 2024-01-04 US claimed
US-20230372316-A1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL-CONTAINING PHARMACEUTICAL COMPOSITION SANTEN PHARMACEUTICAL CO., LTD. (JP) 2023-11-23 US claimed
EP-3320904-B1 PREVENTATIVE AND/OR THERAPEUTIC AGENT CONTAINING PYRIDYL AMINOACETIC ACID COMPOUND FOR TREATING A DISEASE INVOLVING A GREATLY ELEVATED INTRAOCULAR PRESSURE SANTEN PHARMACEUTICAL CO LTD (JP) 2023-07-05 EP claimed
EP-3888654-B1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL CONTAINING PHARMACEUTICAL COMPOSITION SANTEN PHARMACEUTICAL CO LTD (JP) 2023-06-14 EP claimed
US-11331311-B2 Prophylactic and/or therapeutic agent containing pyridylaminoacetic acid compound SANTEN PHARMACEUTICAL CO., LTD. (JP) 2022-05-17 US claimed
US-20220054466-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A PYRIDYLAMINOACETIC ACID COMPOUND SANTEN PHARMACEUTICAL CO., LTD. (JP) 2022-02-24 US claimed
US-20210330654-A1 AGENT FOR TREATING OR PREVENTING GLAUCOMA INCLUDING A SULFONAMIDE COMPOUND AND ANOTHER DRUG SANTEN PHARMACEUTICAL CO., LTD. (JP) 2021-10-28 US claimed
EP-3888654-A1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL CONTAINING PHARMACEUTICAL COMPOSITION Santen Pharmaceutical Co., Ltd. (JP) 2021-10-06 EP claimed
US-20160317512-A1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL-CONTAINING PHARMACEUTICAL COMPOSITION SANTEN PHARMACEUTICAL CO., LTD. (JP) 2016-11-03 US claimed
US-20160228421-A1 COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA COMPRISING A SULFONAMIDE COMPOUND AND ANOTHER DRUG SANTEN PHARMACEUTICAL CO., LTD. (JP) 2016-08-11 US claimed
US-9339496-B2 Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist SANTEN PHARMACEUTICAL CO., LTD. (JP) 2016-05-17 US claimed
EP-2415763-B1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA UBE INDUSTRIES (JP) 2016-01-27 EP claimed
US-8648097-B2 Pyridylaminoacetic acid compound UBE INDUSTRIES, LTD. (JP) 2014-02-11 US claimed
US-20140018396-A1 COMBINATION OF SULFONAMIDE COMPOUND SANTEN PHARMACEUTICAL CO., LTD. (JP) 2014-01-16 US claimed
US-20120190852-A1 MEDICAL COMPOSITION FOR TREATMENT OR PROPHYLAXIS OF GLAUCOMA UBE INDUSTRIES, LTD. (JP) 2012-07-26 US claimed
EP-2476678-A1 SUBSTITUTED CARBONYL COMPOUNDS Ube Industries, Ltd. (JP) 2012-07-18 EP claimed
US-20110054172-A1 PYRIDYLAMINOACETIC ACID COMPOUND UBE CORPORATION (JP) 2011-03-03 US claimed
EP-2264009-A1 PYRIDYLAMINOACETIC ACID COMPOUND Ube Industries, Ltd. (JP) 2010-12-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160317512-A1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL-CONTAINING PHARMACEUTICAL COMPOSITION PAOX, CYP4A11, PAH PTGER2 296/4885PTGER4 237/4885
US-20140018396-A1 COMBINATION OF SULFONAMIDE COMPOUND CHUK, PTGIS, PTGIR PTGER2 58/4885PTGER4 78/4885
US-20160228421-A1 COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA COMPRISING A SULFONAMIDE COMPOUND AND ANOTHER DRUG PTGIS, PTGIR, PTGS1 PTGER2 6/4885PTGER4 25/4885
US-20240024484-A1 PHARMACEUTICAL COMPOSITION CONTAINING PYRIDYLAMINOACETIC ACID COMPOUND AADAT, DDC, PDE12 PTGER2 505/4885PTGER4 567/4885
US-11974994-B2 Agent for treating or preventing glaucoma including a sulfonamide compound and another drug PTGIS, PTGIR, PTGS1 PTGER2 13/4885PTGER4 51/4885
US-20240000763-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A PYRIDYLAMINOACETIC ACID COMPOUND REN, AGTR2, PTGIS PTGER2 314/4885PTGER4 515/4885
US-20230372316-A1 PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL-CONTAINING PHARMACEUTICAL COMPOSITION PAOX, CYP4A11, PAH PTGER2 296/4885PTGER4 237/4885
US-20220054466-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A PYRIDYLAMINOACETIC ACID COMPOUND REN, AGTR2, PTGIS PTGER2 314/4885PTGER4 515/4885
US-11331311-B2 Prophylactic and/or therapeutic agent containing pyridylaminoacetic acid compound AADAC, AADAT, PLPBP PTGER2 1073/4885PTGER4 2062/4885
US-20110054172-A1 PYRIDYLAMINOACETIC ACID COMPOUND PTGER2, PTGER1, PTGDR2 PTGER2 1/4885PTGER4 17/4885
US-20120190852-A1 MEDICAL COMPOSITION FOR TREATMENT OR PROPHYLAXIS OF GLAUCOMA F12, C1S, AKR1C3 PTGER2 24/4885PTGER4 133/4885
US-20210330654-A1 AGENT FOR TREATING OR PREVENTING GLAUCOMA INCLUDING A SULFONAMIDE COMPOUND AND ANOTHER DRUG PTGIS, PTGIR, PTGS1 PTGER2 13/4885PTGER4 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.