SCHEMBL5332673

SCHEMBL5332673

CCS(=O)(=O)c1c(F)cccc1C(=O)N(C)C1(CC2CCOCC2)CCNCC1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.33
CNR2 P34972 7/20 0.33
OPRD1 P41143 3/20 0.33
OPRM1 P35372 1/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 2/20 0.32
HSD11B1 P28845 1/20 0.32
KCNH2 Q12809 2/20 0.31
CYP2D6 P10635 1/20 0.31
OPRL1 P41146 1/20 0.31
REN P00797 1/20 0.31
CXCR2 P25025 1/20 0.30
MEN1 O00255 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134854 0.79 CNR1 (0.37) CNR1CNR2KMT2APOLBKCNH2
SCHEMBL5135170 0.76 OPRM1 (0.39) CNR1CNR2OPRD1OPRM1POLB
SCHEMBL5135169 0.64 PARP1 (0.39) CNR1CNR2OPRM1OPRL1
SCHEMBL5332677 0.64 OPRL1 (0.33) OPRL1
SCHEMBL3614449 0.63 HPGD (0.49) KMT2APOLBHSD11B1CYP2D6MEN1
SCHEMBL5135172 0.62 OPRM1 (0.37) CNR1CNR2OPRM1OPRL1
SCHEMBL1290783 0.61 OPRM1 (0.35) OPRM1KMT2AOPRL1
SCHEMBL12727293 0.59 PKM (0.47) CXCR2
SCHEMBL415193 0.58 CYP2D6 (0.46) POLBSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL5190868 0.58 SLC6A4 (0.45) SLC6A2SLC6A4SLC6A3HSD11B1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed