SCHEMBL5333330

SCHEMBL5333330

C=CCc1c(-c2ccc(N)cc2)ccc(N(CC=C)CC=C)c1CC=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10885447 0.98
SCHEMBL2787924 0.80 ALDH1A1 (0.32)
SCHEMBL6139923 0.78 ALDH1A1 (0.35)
SCHEMBL1334154 0.77 IMPDH2 (0.41)
SCHEMBL29900410 0.70 NCOA1 (0.44)
SCHEMBL29499603 0.68 CASP1 (0.34)
SCHEMBL2221665 0.68 CASP1 (0.34)
SCHEMBL8675962 0.68 GABRA1 (0.44)
Ammonia Solution, Strong SCHEMBL5991120 0.67 CASP1 (0.33)
SCHEMBL127344 0.67 ALDH1A1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918881-B1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND AMIRA MEDICAL (US) 2004-02-11 EP claimed
WO-2000039586-A2 TETRAMETHYLBENZIDINE FORMULATION FOR HORSERADISH PEROXIDASE ENZYME ASSAYS SEDUM LABORATORIES (US) 2000-07-06 WO claimed
EP-0918881-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND Mercury Diagnostics Inc. (US) 1999-06-02 EP claimed
US-5824491-A OXIDASE ENZYME AS ANALYTE ON SUBSTRATE, FORMING PEROXIDE, BENZIDINE DYE PRECURSOR, PEROXIDASE ENZYME WITH ANTIPYRENE COMPOUND MERCURY DIAGNOSTICS, INC. (US) 1998-10-20 US claimed
WO-1997044482-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND MERCURY DIAGNOSTICS INC. (US) 1997-11-27 WO claimed
US-5610026-A OF AN AQUEOUS SOLUTION CONTAINING A TETRAALKYLBENZIDINE OR A SALT THEREOF, A PEROXIDE OR A SYSTEM GENERATING HYDROGEN PEROXIDE AND A BUFFER BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1997-03-11 US claimed
US-5491094-A COLORIMETRIC ANALYSIS INDICATOR 3,3*,5,5*-TETRAALKYLBENZIDINE INDUSTRIAL TEST SYSTEMS, INC. (US) 1996-02-13 US claimed
US-5206150-A Tetramethylbenzidine, peroxide and bacitracin as stabilizer; incubation UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1993-04-27 US claimed
EP-0224813-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY WITH A STABILIZER, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-09-26 EP claimed
EP-0224210-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-08-29 EP claimed
US-4891314-A STORAGE STABILITY BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1990-01-02 US claimed
US-4562148-A IMMUNOASSAY, CARBOXYLATE OR SULFONATE POLYMER MILES LABORATORIES, INC. (US) 1985-12-31 US claimed
JP-1104196-A None JP disclosed
JP-8080199-A None JP disclosed
JP-61052300-A None JP disclosed
JP-8313525-A None JP disclosed
US-4385114-A DETERMINATION OF HYDROGEN PEROXIDE OR PEROXIDASE BOEHRINGER MANNHEIM GMBH (DE) 1983-05-24 US disclosed
EP-0078965-A1 Method for preparing an analytical element preventing reagent migration MILES LABORATORIES, INC. (US) 1983-05-18 EP disclosed
EP-0071934-A1 Method for preparing a color stable chromogenic analytical element MILES LABORATORIES, INC. (US) 1983-02-16 EP disclosed
US-4361648-A POLYMERIC MORDANT, TETRAALKYLBENZIDINE HYDROCHLORIDE, ENZYME, PEROXIDATIVELY ACTIVE MATERIAL MILES LABORATORIES, INC. (US) 1982-11-30 US disclosed