SCHEMBL5335642

SCHEMBL5335642

NC(=O)c1ccc(-c2ccccc2)c(N2C=CON2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 7/20 0.40
ALDH1A1 P00352 1/20 0.40
MKNK1 Q9BUB5 5/20 0.38
MKNK2 Q9HBH9 4/20 0.37
IP6K1 Q92551 1/20 0.36
JAK3 P52333 3/20 0.36
JAK2 O60674 2/20 0.36
JAK1 P23458 2/20 0.36
TYK2 P29597 2/20 0.36
CDC7 O00311 1/20 0.36
PLK4 O00444 1/20 0.36
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
MAPK13 O15264 1/20 0.36
PDPK1 O15530 1/20 0.36
DYRK3 O43781 1/20 0.36
ROCK2 O75116 1/20 0.36
RPS6KA5 O75582 1/20 0.36
PRKD3 O94806 1/20 0.36
PAK4 O96013 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5420145 0.78 MKNK1 (0.38) CHEK2ALDH1A1MKNK1MKNK2IP6K1
SCHEMBL7680894 0.73 BCAT2 (0.50) BCAT2DHODH
SCHEMBL7680902 0.73 BCAT2 (0.40) AURKABCAT2DHODH
SCHEMBL7673605 0.71 PARP10 (0.37) ALDH1A1MKNK1MKNK2BCAT2
SCHEMBL30556675 0.71 HTR6 (0.58) ALDH1A1PRKD2
SCHEMBL2026663 0.70 L3MBTL1 (0.52) CHEK2MKNK1MKNK2IP6K1JAK3
SCHEMBL30903715 0.70 L3MBTL1 (0.52) CHEK2MKNK1MKNK2IP6K1JAK3
SCHEMBL28218967 0.70 PTGS1 (0.51) CHEK2ALDH1A1MKNK1MKNK2BCAT2
Hydrochloric Acid SCHEMBL28812686 0.69 CHEK2 (0.50) CHEK2MKNK1MKNK2IP6K1JAK3
SCHEMBL3781170 0.68 MKNK1 (0.53) CHEK2ALDH1A1MKNK1MKNK2IP6K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007077457-A9 TREATMENT OF EQUINE LAMINITIS WITH 5-HT1B/ 1D ANTAGONISTS ROYAL VETERINARY COLLEGE (GB) 2007-10-18 WO claimed
WO-2007077457-A2 TREATMENT OF EQUINE LAMINITIS WITH 5-HT1B/ 1D ANTAGONISTS THE ROYAL VETERINARY COLLEGE (GB) 2007-07-12 WO claimed
WO-2007077457-A9 TREATMENT OF EQUINE LAMINITIS WITH 5-HT1B/ 1D ANTAGONISTS ROYAL VETERINARY COLLEGE (GB) 2007-10-18 WO disclosed