SCHEMBL7680902

SCHEMBL7680902

NC(=O)c1cccc(N2C=CON2)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.40
PARP1 P09874 6/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
NPC1 O15118 2/20 0.35
DHODH Q02127 1/20 0.35
IKBKB O14920 2/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
MAP2 P11137 2/20 0.34
AURKA O14965 1/20 0.34
BRD4 O60885 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2283018 0.83 NPC1 (0.44) BCAT2PARP1NPC1SIRT1AURKA
SCHEMBL7680894 0.79 BCAT2 (0.50) BCAT2PARP1KEAP1NFE2L2NPC1
SCHEMBL2487391 0.77 ALDH1A1 (0.47)
SCHEMBL21801994 0.73
SCHEMBL2789494 0.73 ALDH1A1 (0.42)
SCHEMBL5335642 0.73 CHEK2 (0.40) BCAT2DHODHAURKA
SCHEMBL27214460 0.73 BCAT2 (0.63) BCAT2PARP1KEAP1NFE2L2DHODH
SCHEMBL7676034 0.71 MEN1 (0.39)
SCHEMBL379430 0.70 HTR6 (0.51) PARP1NPC1
SCHEMBL7680897 0.70 ALDH1A1 (0.51) BCAT2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6369088-B2 ANTIDIABETIC AGENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-04-09 US disclosed