SCHEMBL5339211

SCHEMBL5339211

CCN1C(=O)NC(c2cccc(OC)c2)C(C(=O)O)=C1C

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
TDP1 Q9NUW8 2/20 0.58
HTT P42858 1/20 0.53
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
LMNA P02545 5/20 0.49
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TSHR P16473 1/20 0.47
TRPC5 Q9UL62 1/20 0.47
APOBEC3A P31941 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14413854 0.76 NPSR1 (0.69) ALDH1A1HTT
SCHEMBL19732952 0.76 NPSR1 (0.69) ALDH1A1HTT
SCHEMBL4425507 0.73 LMNA (0.39) ALDH1A1LMNARECQLMEN1KMT2A
SCHEMBL6609319 0.70 ALDH1A1 (0.46) ALDH1A1CYP2C9
SCHEMBL3395610 0.70 KIF11 (0.75) ALDH1A1SMN1; SMN2TSHR
SCHEMBL19752619 0.70 KIF11 (0.75) ALDH1A1SMN1; SMN2TSHR
SCHEMBL10564440 0.68 CACNA1F (0.61) ALDH1A1
SCHEMBL8030679 0.68 DRD2 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL13425599 0.68 TP53 (0.50) ALDH1A1LMNA
SCHEMBL10113323 0.67 KMT2A (0.74) ALDH1A1HTTLMNASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007101213-A2 NOVEL 2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINES, BICYCLIC PYRIMIDINE DIONES AND IMIDAZOLIDINE-2,4-DIONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2007-09-07 WO disclosed