SCHEMBL534317

SCHEMBL534317

O=C(O)N1CCCC(c2ccc(-c3ccc(-c4cc(F)cc(F)c4)cc3CO)cc2Cl)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 9/20 0.41
FFAR2 O15552 1/20 0.35
GRM5 P41594 1/20 0.34
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
EPHX2 P34913 2/20 0.33
OPRL1 P41146 1/20 0.33
HSD11B1 P28845 1/20 0.33
PTGDR Q13258 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL556088 0.74 REN (0.41) FFAR2
SCHEMBL28264816 0.68 PROKR1 (0.38) PROKR1ALDH1A1
SCHEMBL4392361 0.67 KMT2A (0.41) PROKR1ALDH1A1MEN1KMT2AEPHX2
SCHEMBL4754555 0.66 PROKR1 (0.48) PROKR1OPRL1
SCHEMBL2364516 0.62 GRM5 (0.44) GRM5ALDH1A1MEN1KMT2AOPRL1
SCHEMBL19212445 0.62 GRM5 (0.48) GRM5KMT2AEPHX2OPRL1
SCHEMBL4099888 0.62 RAB9A (0.57) PROKR1GRM5ALDH1A1HSD11B1
SCHEMBL3999994 0.61 SLC6A2 (0.57) PROKR1HSD11B1
SCHEMBL3410172 0.61 PROKR1 (0.38) PROKR1ALDH1A1
Bicarbonate SCHEMBL17644401 0.60 OPRL1 (0.51) PROKR1GRM5OPRL1PTGDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed