SCHEMBL5352932

SCHEMBL5352932

CNC(=O)Cc1ccc(C2=C(C(=O)O)N3C(=O)[C@H]([C@@H](C)O[Si](C)(C)C)[C@H]3C2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.34
FAAH O00519 3/20 0.34
HDAC4 P56524 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
ELANE P08246 1/20 0.32
MAPT P10636 2/20 0.31
CASP1 P29466 1/20 0.31
CASP3 P42574 1/20 0.31
POLB P06746 1/20 0.31
PKM P14618 1/20 0.31
HTT P42858 1/20 0.31
DUSP3 P51452 1/20 0.31
PTPN5 P54829 1/20 0.31
PTPN11 Q06124 1/20 0.31
ESR1 P03372 1/20 0.31
CHRM1 P11229 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5338872 0.90 KDM4E (0.36) MAPK1FAAHKDM4ELMNAESR1
SCHEMBL5342069 0.89 MAPK1 (0.34) MAPK1FAAHTDP1KDM4ELMNA
SCHEMBL5353135 0.88 RAB9A (0.41) FAAHKDM4ELMNAALDH1A1HPGD
SCHEMBL5340966 0.87 CYP2D6 (0.35) KDM4ELMNAELANEESR1CHRM1
SCHEMBL14517752 0.87 FAAH (0.33) FAAHHDAC4ELANE
SCHEMBL5336434 0.86 KDM4E (0.42) MAPK1HDAC4TDP1KDM4ELMNA
SCHEMBL5353271 0.84 LMNA (0.34) KDM4ELMNAELANEESR1CHRM1
SCHEMBL5340133 0.84 ADAMTS4 (0.35) KDM4ELMNAMAPTESR1CHRM1
SCHEMBL5344996 0.82 SYK (0.39) LMNAHTT
SCHEMBL5344796 0.81 BCL2 (0.34) KDM4ELMNAESR1CHRM1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205291-B2 High mouth absorption; antibiotics against gramnegative, grampositive bacteria espscially Staphlococcus pneumonia, Hemophilus influenza DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2007-04-17 US disclosed
US-20050020566-A1 Novel carbapenem compounds DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2005-01-27 US disclosed
EP-1443047-A1 NOVEL CARBAPENEM COMPOUNDS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2004-08-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020566-A1 Novel carbapenem compounds HPN, PRSS1, BPGM MAPK1 3834/4885FAAH 4701/4885HDAC4 2091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.