SCHEMBL5357212

SCHEMBL5357212

N#Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nc1CO

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.34
NPSR1 Q6W5P4 2/20 0.33
MAOA P21397 1/20 0.32
STAT3 P40763 1/20 0.32
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 3/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
ALOX12 P18054 1/20 0.30
KCNN4 O15554 1/20 0.30
KCNA3 P22001 1/20 0.30
AURKA O14965 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360814 0.85 TSHR (0.34) TSHRNPSR1ALDH1A1MEN1KMT2A
SCHEMBL11553962 0.72 SMN1; SMN2 (0.43) TSHRRAB9ANPC1ALDH1A1MEN1
SCHEMBL5353528 0.71 MAPT (0.43) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL5363475 0.71 KDM4E (0.48) NPSR1RAB9ANPC1ALDH1A1MEN1
SCHEMBL5357402 0.66 P2RX7 (0.40) TSHRNPSR1MAOARAB9AALDH1A1
SCHEMBL27815941 0.66 PTGER1 (0.40) TSHRNPSR1RAB9ANPC1ALDH1A1
SCHEMBL4369849 0.66 ALDH1A1 (0.35) TSHRNPSR1RAB9ANPC1ALDH1A1
SCHEMBL3147317 0.66 GABRP (0.40) ALDH1A1TDP1KDM4ELMNA
SCHEMBL27865251 0.65 AURKA (0.41) TSHRNPSR1MAOARAB9AMEN1
SCHEMBL5366279 0.65 KDM4E (0.34) ALDH1A1TDP1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed