SCHEMBL5362014

SCHEMBL5362014

CC(C)OCCNC(=O)c1ccc2ncc3nncn3c2c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PAX8 Q06710 1/20 0.43
NAMPT P43490 5/20 0.42
LMNA P02545 1/20 0.41
HPGD P15428 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5358234 0.91 LMNA (0.48) LMNAHPGDCYP1A2CYP2C9MAPK1
SCHEMBL5355346 0.82 LMNA (0.55) ALDH1A1LMNAHPGDCYP1A2CYP2C9
SCHEMBL5364346 0.80 TP53 (0.52) ALDH1A1NAMPTLMNAHPGDKMT2A
SCHEMBL5352150 0.77 ALDH1A1 (0.55) ALDH1A1HPGDCYP1A2CYP2C9MAPK1
SCHEMBL5358019 0.75 FGFR1 (0.49) ALDH1A1L3MBTL1LMNAHPGDMAPK1
SCHEMBL31744961 0.74 FGFR1 (0.40) ALDH1A1NAMPTLMNAHPGDMAPK1
SCHEMBL5356306 0.73 KMT2A (0.54) ALDH1A1TSHRHPGDCYP1A2CYP2C9
SCHEMBL13681674 0.69 HTT (0.74) L3MBTL1NAMPTLMNAMAPK1KMT2A
SCHEMBL5426958 0.68 GSK3B (0.64) ALDH1A1TSHRL3MBTL1NAMPTKMT2A
SCHEMBL13450223 0.67 EPHX2 (0.59) ALDH1A1TSHRL3MBTL1PAX8NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202245-B2 Substituted 4-amino[1,2,4]triazolo[4,3-a] quinoxalines PFIZER INC. (US) 2007-04-10 US disclosed