Adenosine

Adenosine

SCHEMBL536558

Nc1ncnc2[nH]cnc12.Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3

The experimentally established mechanism targets of Adenosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 known ✓ P0DMS8 4/20 0.81
ADORA2A known ✓ P29274 1/20 0.81
ADORA2B known ✓ P29275 1/20 0.81
ADORA1 known ✓ P30542 1/20 0.81
DOT1L Q8TEK3 2/20 0.81
DPP4 P27487 1/20 0.81
MEN1 O00255 1/20 0.81
SLC28A1 O00337 1/20 0.81
MAP3K7 O43318 1/20 0.81
SLC28A2 O43868 1/20 0.81
GAPDH P04406 1/20 0.81
MAPK1 P28482 1/20 0.81
STAT6 P42226 1/20 0.81
PI4KA P42356 1/20 0.81
KMT2A Q03164 1/20 0.81
SMN1; SMN2 Q16637 1/20 0.81
PI4K2B Q8TCG2 1/20 0.81
SLC29A1 Q99808 1/20 0.81
PI4K2A Q9BTU6 1/20 0.81
SLC28A3 Q9HAS3 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Vidarabine SCHEMBL27371675 1.00 ADORA3 (0.81) ADORA3DOT1LDPP4MEN1SLC28A1
Inosine SCHEMBL21840403 0.94 ADORA3 (0.72) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL23201584 0.92 ADORA3 (0.68) ADORA3DOT1LDPP4MEN1SLC28A1
Vidarabine SCHEMBL27261659 0.92 ADORA3 (0.71) ADORA3DOT1LDPP4MEN1SLC28A1
Vidarabine SCHEMBL27261788 0.91 ADORA3 (0.70) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL23804425 0.90 ADORA3 (1.00) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL1821276 0.90 ADORA3 (1.00) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL24538665 0.90 ADORA3 (1.00) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL2228590 0.90 ADORA3 (1.00) ADORA3DOT1LDPP4MEN1SLC28A1
Adenosine SCHEMBL406207 0.90 ADORA3 (1.00) ADORA3DOT1LDPP4MEN1SLC28A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118058376-A Two-way solid-state fermentation ginseng sweet potato preserved fruit with ganoderma lucidum and preparation method thereof 吉林省养易多科技有限公司 2024-05-24 CN disclosed
US-11905308-B2 Nucleic acid compound and oligonucleotide OSAKA UNIVERSITY (JP) 2024-02-20 US disclosed
CN-115521245-B Alkaloid compound in purslane, and extraction and separation method and application thereof 辽宁中医药大学 2024-01-19 CN disclosed
CN-113698446-B Alkaloid compound in purslane and extraction and separation method thereof 辽宁中医药大学 2023-05-16 CN disclosed
CN-114213473-B Three alkaloid compounds in purslane and extraction and separation method thereof 辽宁中医药大学 2023-04-25 CN disclosed
US-20230100842-A1 TRIAZOLO[4,5-D] PYRAMIDINE DERIVATIVES AND THEIR USE AS PURINE RECEPTOR ANTAGONISTS LIGAND UK DEVELOPMENT LIMITED (GB) 2023-03-30 US disclosed
CN-115521245-A Alkaloid compound in purslane and extraction and separation method and application thereof 辽宁中医药大学 2022-12-27 CN disclosed
US-20220169671-A1 NUCLEIC ACID COMPOUND AND OLIGONUCLEOTIDE OSAKA UNIVERSITY (JP) 2022-06-02 US disclosed
CN-113264828-B Benzoic acid compound in purslane and extraction and separation method thereof 辽宁中医药大学 2022-05-17 CN disclosed
CN-114213473-A Three alkaloid compounds in purslane and extraction and separation method thereof 辽宁中医药大学 2022-03-22 CN disclosed
US-6197788-B1 (−)-mefloquine to block puringergic receptors and to treat movement or neurodegenerative disorders VERNALIS RESEARCH LIMITED (GB) 2001-03-06 US disclosed
WO-2001002409-A1 THIENO- AND FUROPYRIMIDINE DERIVATIVES AS A2A-RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-01-11 WO disclosed
WO-2000013682-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS.(II) VERNALIS RESEARCH LIMITED (GB) 2000-03-16 WO disclosed
WO-2000013681-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS (I) VERNALIS RESEARCH LIMITED (GB) 2000-03-16 WO disclosed
EP-0975345-A1 (-)-MEFLOQUINE TO BLOCK PURINERGIC RECEPTORS AND TO TREAT MOVEMENT OR NEURODEGENERATIVE DISORDERS Cerebrus Pharmaceuticals Limited (GB) 2000-02-02 EP disclosed
WO-1999026627-A1 (-)-MEFLOQUINE TO BLOCK PURINERGIC RECEPTORS AND TO TREAT MOVEMENT OR NEURODEGENERATIVE DISORDERS CEREBRUS LIMITED (GB) 1999-06-03 WO disclosed
EP-0420977-A4 NOVEL LYOPHILIZED AND RECONSTITUTED RED BLOOD CELL COMPOSITIONS 1991-11-06 EP disclosed
EP-0420977-A1 NOVEL LYOPHILIZED AND RECONSTITUTED RED BLOOD CELL COMPOSITIONS CRYOPHARM CORPORATION (US) 1991-04-10 EP disclosed
WO-1990012582-A1 NOVEL LYOPHILIZED AND RECONSTITUTED RED BLOOD CELL COMPOSITIONS CRYOPHARM CORPORATION (US) 1990-11-01 WO disclosed
US-4354913-A MEMBRANE HAVING SURFACE CONTAINING THE REACTION PRODUCT OF GLUTARALDEHYDE AND THE ENZYME RADELKIS ELEKTROKEMIAI MUSZERGYARTO SZOVETKEZET (HU) 1982-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11905308-B2 Nucleic acid compound and oligonucleotide NSUN2, NUDT1, EFTUD2 ADORA3 348/4885ADORA2A 493/4885ADORA2B 565/4885
US-20220169671-A1 NUCLEIC ACID COMPOUND AND OLIGONUCLEOTIDE NSUN2, NUDT1, EFTUD2 ADORA3 348/4885ADORA2A 493/4885ADORA2B 565/4885
US-20230100842-A1 TRIAZOLO[4,5-D] PYRAMIDINE DERIVATIVES AND THEIR USE AS PURINE RECEPTOR ANTAGONISTS P2RX5, P2RY1, P2RX3 ADORA3 14/4885ADORA2A 11/4885ADORA2B 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.