SCHEMBL5368699

SCHEMBL5368699

N#Cc1ccccc1Oc1cc(Cc2ccc(=O)[nH]n2)ccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 13/20 0.39
CYP3A4 P08684 1/20 0.36
SLC22A12 Q96S37 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
AKR1B1 P15121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5382509 0.85 CYP3A4 (0.42) CYP3A4SLC22A12PRMT5WDR77
SCHEMBL5374946 0.85 CYP3A4 (0.42) ARCYP3A4PRMT5WDR77AKR1B1
SCHEMBL5366909 0.83 CYP3A4 (0.46) CYP3A4AKR1B1
SCHEMBL5373732 0.82 CYP3A4 (0.45) ARCYP3A4PRMT5WDR77
SCHEMBL5375034 0.82 CYP3A4 (0.37) ARCYP3A4SLC22A12
SCHEMBL5377568 0.77 CYP3A4 (0.47) ARCYP3A4
SCHEMBL5374482 0.77 CYP3A4 (0.61) ARCYP3A4PRMT5WDR77AKR1B1
SCHEMBL5370291 0.73 CYP3A4 (0.43) CYP3A4SLC22A12AKR1B1
SCHEMBL5365226 0.73 SLC22A12 (0.40) ARCYP3A4SLC22A12
SCHEMBL5377392 0.73 CYP3A4 (0.39) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed