Reserpine

Reserpine

SCHEMBL5372168

COC(=O)C1C2CC3c4[nH]c5cc(OC)ccc5c4CCN3CC2CC(OC(=O)c2cc(OC)c(OC)c(OC)c2)C1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC18A2

The experimentally established mechanism targets of Reserpine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A2 known ✓ Q05940 1/20 1.00
MEN1 O00255 13/20 1.00
KMT2A Q03164 13/20 1.00
KDM4E B2RXH2 9/20 1.00
TDP1 Q9NUW8 7/20 1.00
TSHR P16473 6/20 1.00
HBB P68871 5/20 1.00
MAPT P10636 5/20 1.00
CYP3A4 P08684 4/20 1.00
ALDH1A1 P00352 4/20 1.00
USP2 O75604 4/20 1.00
CASP1 P29466 4/20 1.00
ALOX15 P16050 4/20 1.00
KCNH2 Q12809 3/20 1.00
CASP7 P55210 3/20 1.00
HSD17B10 Q99714 3/20 1.00
ADORA3 P0DMS8 2/20 1.00
OPRM1 P35372 2/20 1.00
OPRK1 P41145 2/20 1.00
CYP1A2 P05177 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Reserpine SCHEMBL20402680 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL15385127 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Isoreserpine SCHEMBL731599 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL1172973 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL4562878 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL12732449 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL8262666 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL14379427 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL5372164 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL22002247 1.00 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7241797-B2 Method of increasing milk production UNIVERSITY OF CINCINNATI (US) 2007-07-10 US claimed
US-20030139420-A1 Method of increasing milk production NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-07-24 US claimed
EP-0652767-B1 TREATMENT OF HUMAN LACTATION FAILURE PHARMACIA & UPJOHN AB (SE) 1999-09-15 EP claimed
US-5276014-A Human growth factor KABI PHARMACIA AB (SE) 1994-01-04 US claimed
US-20230301984-A1 CYCLIC COMPOUNDS FOR USE IN TREATING RETINAL DEGENERATION THE USA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2023-09-28 US disclosed
EP-4175636-A2 CYCLIC COMPOUNDS FOR USE IN TREATING RETINAL DEGENERATION The United States of America, as represented by the Secretary, Department of Health and Human Services (US) 2023-05-10 EP disclosed
EP-3837229-B1 METHOD FOR MANUFACTURING A CONSOLIDATED DENSIFIED PART FROM CERAMIC OR CARBON COMMISSARIAT ENERGIE ATOMIQUE (FR) 2022-06-22 EP disclosed
WO-2022006439-A2 COMPOUND EMBODIMENTS FOR TREATING RETINAL DEGENERATION AND METHOD EMBODIMENTS OF MAKING AND USING THE SAME THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2022-01-06 WO disclosed
US-20210360924-A1 PLANT OR SEED COATING UNIV SOUTHAMPTON (GB) 2021-11-25 US disclosed
EP-3837229-A1 METHOD FOR MANUFACTURING A CONSOLIDATED DENSIFIED PART FROM CERAMIC OR CARBON Commissariat à l'énergie atomique et aux énergies alternatives (FR) 2021-06-23 EP disclosed
WO-2020058647-A1 METHOD FOR MANUFACTURING A CONSOLIDATED DENSIFIED PART FROM CERAMIC OR CARBON COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2020-03-26 WO disclosed
US-9012838-B2 Covalently functionalized nanodiamond-based MALDI matrices and methods of use thereof UNIVERSITY OF SASKATCHEWAN (CA) 2015-04-21 US disclosed
US-20080267948-A1 Croos-B Structure Binding Compounds CROSSBETA BIOSCIENCES B.V. (NL) 2008-10-30 US disclosed
US-7241797-B2 Method of increasing milk production UNIVERSITY OF CINCINNATI (US) 2007-07-10 US disclosed
US-20030139420-A1 Method of increasing milk production NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-07-24 US disclosed
EP-0652767-B1 TREATMENT OF HUMAN LACTATION FAILURE PHARMACIA & UPJOHN AB (SE) 1999-09-15 EP disclosed
US-5276014-A Human growth factor KABI PHARMACIA AB (SE) 1994-01-04 US disclosed
US-4298611-A ADMINISTERING 2-CHLORO-6-METHYLERGOLINE-8-BETA-ACETONITRILE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1981-11-03 US disclosed
EP-0005074-A1 A material and composition for reducing blood pressure MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1979-10-31 EP disclosed
EP-0005057-A1 A material and composition for reducing blood pressure MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1979-10-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080267948-A1 Croos-B Structure Binding Compounds CACYBP, TBCB, MYCBP SLC18A2 2613/4885MEN1 4546/4885KMT2A 4555/4885
US-20230301984-A1 CYCLIC COMPOUNDS FOR USE IN TREATING RETINAL DEGENERATION ALDH1A2, PDE6D, PDE6C SLC18A2 916/4885MEN1 4843/4885KMT2A 1905/4885
US-20210360924-A1 PLANT OR SEED COATING PNMT, TPH1, TPH2 SLC18A2 49/4885MEN1 3232/4885KMT2A 2561/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.