SCHEMBL5387953

SCHEMBL5387953

CC(=O)OCc1nc2cccc(N3CCN(C(=O)O)CC3)c2n1C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 1/20 0.38
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HTR7 P34969 3/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRM2 Q14416 1/20 0.34
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4163673 0.88 ACHE (0.42) ALDH1A1MAPTGAASMN1; SMN2
SCHEMBL5549018 0.85 NCF1 (0.39) NCF1ALDH1A1MAPTGAASMN1; SMN2
SCHEMBL5547464 0.83 SLC6A7 (0.34) ALDH1A1CYP1A2CYP2C19GRM2HTR1A
SCHEMBL4885947 0.78 HTR1A (0.38) ALDH1A1MAPTTMEM97SIGMAR1HTR1A
SCHEMBL4178891 0.74 CKS1B (0.43) ALDH1A1MAPT
SCHEMBL4889066 0.72 HTR7 (0.44) MAPTMEN1KMT2AHTR7HTR1A
SCHEMBL4887206 0.72 BACE1 (0.51) MAPTMEN1KMT2A
SCHEMBL4878710 0.71 ACHE (0.42) ALDH1A1MAPTGAASMN1; SMN2
SCHEMBL5549046 0.69 KDM4E (0.35) ALDH1A1MAPTSMN1; SMN2KMT2AHTR7
SCHEMBL4889339 0.68 SLC6A7 (0.34) ALDH1A1MAPTGRM2HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789045-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-30 EP disclosed
WO-2006023400-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-03-02 WO disclosed