SCHEMBL5409102

SCHEMBL5409102

O=C(O)CCN(CCc1ccncc1)C(=O)c1ccccc1-c1ccccc1C(=O)NCc1c(F)cccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK1 P28482 1/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MAPK14 Q16539 3/20 0.38
MAPK7 Q13164 2/20 0.38
POLB P06746 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
USP2 O75604 1/20 0.36
DNMT3B Q9UBC3 1/20 0.36
ROCK2 O75116 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5409280 0.93 RAB9A (0.44) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5399560 0.91 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5394224 0.90 HTT (0.50) ALDH1A1MAPK1KMT2AHTTUSP2
SCHEMBL5395784 0.89 ALDH1A1 (0.43) ALDH1A1KMT2ANPC1RAB9AMAPK14
SCHEMBL5402400 0.88 RAB9A (0.44) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5397914 0.88 MAPK1 (0.49) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5399511 0.88 KMT2A (0.48) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5392177 0.87 AURKA (0.44) ALDH1A1SMN1; SMN2MAPK1KMT2AHTT
SCHEMBL5403086 0.86 KCNK3 (0.46) ALDH1A1KMT2ARAB9APOLBHDAC1
SCHEMBL5403388 0.86 LMNA (0.48) ALDH1A1SMN1; SMN2KMT2AHTTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB ALDH1A1 1256/4885SMN1; SMN2 57/4885MAPK1 1369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.