SCHEMBL5457191

SCHEMBL5457191

CN1CCc2cc(N(C)C)c(S(=O)(=O)c3ccc(Cc4cccc(OC(F)(F)F)c4)cc3)cc2CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 3/20 0.38
PRMT6 Q96LA8 3/20 0.38
HTR2A P28223 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
HRH3 Q9Y5N1 1/20 0.37
TBXA2R P21731 1/20 0.36
PTGDR Q13258 1/20 0.36
KDM2B Q8NHM5 1/20 0.36
LTA4H P09960 1/20 0.36
GPR52 Q9Y2T5 1/20 0.35
CHRM5 P08912 1/20 0.35
NR3C1 P04150 1/20 0.35
CNR2 P34972 1/20 0.35
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5453022 0.92 HTR2A (0.46) HTR2ASLC6A4SLC6A3HRH3KDM2B
SCHEMBL5448126 0.89 LTA4H (0.47) HRH3LTA4H
SCHEMBL5451428 0.86 GALR3 (0.42) CARM1PRMT6HTR2AGPR52
SCHEMBL5466786 0.85 SIGMAR1 (0.42) HTR2ASLC6A4SLC6A3
SCHEMBL14411990 0.84 HTR6 (0.43) HTR2ACHRM2CHRM1HRH3LTA4H
SCHEMBL5455402 0.84 HRH3 (0.38) HTR2AHRH3
SCHEMBL5458151 0.83 LTA4H (0.43) HTR2ALTA4H
SCHEMBL5459209 0.81 DRD1 (0.43) HTR2ASLC6A4SLC6A3LTA4HCNR2
SCHEMBL5445721 0.81 USP2 (0.41) HTR2A
SCHEMBL5450383 0.81 UTS2R (0.38) HTR2ALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070225276-A1 7-Phenylsulfonyl-Tetrahydro-3-Benzazepine Dervatives as Antipsychotic Agents GLAXO GROUP LIMITED (GB) 2007-09-27 US claimed
US-20070225276-A1 7-Phenylsulfonyl-Tetrahydro-3-Benzazepine Dervatives as Antipsychotic Agents GLAXO GROUP LIMITED (GB) 2007-09-27 US disclosed
EP-1687005-A1 7-PHENYLSULFONYL-TETRAHYDRO-3-BENZAZEPINE DERIVATIVES AS ANTIPSYCHOTIC AGENTS GLAXO GROUP LIMITED (GB) 2006-08-09 EP disclosed
WO-2005051398-A1 7-PHENYLSULFONYL-TETRAHYDRO-3-BENZAZEPINE DERIVATIVES AS ANTIPSYCHOTIC AGENTS GLAXO GROUP LIMITED (GB) 2005-06-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070225276-A1 7-Phenylsulfonyl-Tetrahydro-3-Benzazepine Dervatives as Antipsychotic Agents HTR4, DRD4, SLC6A3 CARM1 598/4885PRMT6 1136/4885HTR2A 448/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.