Hydroxyphenamate

Hydroxyphenamate

SCHEMBL546919

CCC(O)(COC(N)=O)c1ccccc1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
CYP1A2 P05177 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP2D6 P10635 1/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KCNN4 O15554 3/20 0.41
LMNA P02545 2/20 0.40
HSD17B10 Q99714 1/20 0.40
CHRM3 P20309 3/20 0.39
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHRM4 P08173 1/20 0.38
KIF11 P52732 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxyphenamate SCHEMBL5704281 1.00 KMT2A (0.42) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6
SCHEMBL4590400 0.77 MAPT (0.50) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6
SCHEMBL5898588 0.77 MAPT (0.46) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6
Urethane SCHEMBL27979330 0.77 ALOX15 (0.50) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6
SCHEMBL10815680 0.75 CA2 (0.43) CYP1A2KCNN4CHRM3CYP2C9CYP2C19
SCHEMBL4307361 0.75 CYP2C19 (0.56) KMT2ACYP1A2SMN1; SMN2CYP2D6KCNN4
SCHEMBL5898545 0.75 MAPT (0.43) KMT2AMAPTCYP1A2CYP2D6KCNN4
SCHEMBL5704134 0.74 LMNA (0.42) KMT2ACYP1A2SMN1; SMN2LMNACHRM3
SCHEMBL7216196 0.74 NPSR1 (0.44) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6
Urethane SCHEMBL3680047 0.74 ALOX15 (0.56) KMT2AMAPTCYP1A2SMN1; SMN2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 386 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016196726-A9 ANTI-TAU ANTIBODIES AND METHODS OF USE GENENTECH, INC. (US) 2017-04-13 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-8110569-B2 Enantiomerically pure S-etifoxine, pharmaceutical compositions thereof and methods of their use THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-02-07 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-2007741-A1 ENANTIOMERICALLY PURE S-ETIFOXINE, PHARMACEUTICAL COMPOSITIONS THEREOF AND METHODS OF THEIR USE Xytis Inc. (US) 2008-12-31 EP claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
US-20080038331-A1 Enantiomerically pure S-etifoxine, pharmaceutical compositions thereof and methods of their use ANVYL LLC 2008-02-14 US claimed
US-20080039453-A1 Enantiomerically pure R-etifoxine, pharmaceutical compositions thereof and methods of their use OXFORD FINANCE CORPORATION 2008-02-14 US claimed
WO-2007109288-A2 ENANTIOMERICALLY PURE R-ETIFOXINE, PHARMACEUTICAL COMPOSITIONS THEREOF AND METHODS OF THEIR USE XYTIS INC. (US) 2007-09-27 WO claimed
WO-2007109289-A1 ENANTIOMERICALLY PURE S-ETIFOXINE, PHARMACEUTICAL COMPOSITIONS THEREOF AND METHODS OF THEIR USE XYTIS INC. (US) 2007-09-27 WO claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080038331-A1 Enantiomerically pure S-etifoxine, pharmaceutical compositions thereof and methods of their use PYGB, CYP2C9, CYP3A5 KMT2A 1976/4885MAPT 665/4885CYP1A2 60/4885
US-20080039453-A1 Enantiomerically pure R-etifoxine, pharmaceutical compositions thereof and methods of their use PYGB, GRIK5, CYP3A5 KMT2A 1795/4885MAPT 632/4885CYP1A2 69/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.