SCHEMBL5485436

SCHEMBL5485436

N#Cc1ccccc1S(=O)(=O)N1CCOC(CNC(=O)[C@@H](CC2CCCCC2)c2ccc3ccccc3c2C(N)=O)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.38
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
MMP8 P22894 1/20 0.34
MMP13 P45452 1/20 0.34
NPY5R Q15761 1/20 0.33
CNR1 P21554 4/20 0.33
EPHX2 P34913 1/20 0.33
REN P00797 1/20 0.33
KMT2A Q03164 2/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484032 0.81 RAB9A (0.41) ATMALDH1A1CNR1RENRAB9A
SCHEMBL4178441 0.80 CTSL (0.47) ATMKMT2ARAB9A
SCHEMBL4188282 0.79 CTSS (0.54) ATMKMT2A
SCHEMBL4185689 0.77 ATM (0.42) ATMALDH1A1MMP1MMP2MMP3
SCHEMBL4185692 0.77 CTSL (0.45) ATMALDH1A1RENRAB9A
SCHEMBL4191791 0.77 CTSB (0.42) ATMREN
SCHEMBL5490202 0.76 ATM (0.37) ATMTP53TSHRMAPK1HSD17B10
SCHEMBL4181130 0.75 CTSS (0.48) ATMALDH1A1MMP1MMP2MMP3
SCHEMBL4185666 0.74 ATM (0.47) ATMTP53TSHRMAPK1HSD17B10
SCHEMBL4183323 0.73 TSHR (0.44) ATMALDH1A1TP53TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869026-A1 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2007-12-26 EP disclosed
WO-2006105475-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO disclosed