SCHEMBL5490202

SCHEMBL5490202

CCC[C@H](C(=O)NCC1CN(S(=O)(=O)c2ccccc2C#N)CCO1)c1ccccc1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RAB9A P51151 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TSHR P16473 2/20 0.34
CTSS P25774 2/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ACLY P53396 1/20 0.33
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
GAA P10253 1/20 0.33
KDM2B Q8NHM5 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5487435 0.80 CTSL (0.40) ATMKDM4ERAB9ACTSSMAPK1
Hydrochloric Acid SCHEMBL4189192 0.79 ATM (0.40) ATMKDM4EPKMCTDSP1TDP1
SCHEMBL4185666 0.79 ATM (0.47) ATMKDM4EPKMCTDSP1TDP1
SCHEMBL4188373 0.77 CTSS (0.39) ATMKDM4ERAB9ACTSSMAPK1
SCHEMBL5485436 0.76 ATM (0.38) ATMRAB9AJAK2JAK1TSHR
SCHEMBL5484026 0.76 MAPK1 (0.47) ATMRAB9AMAPK1
SCHEMBL4171001 0.76 ATM (0.41) ATMKDM4ERAB9ATSHRTP53
SCHEMBL4175687 0.76 CNR1 (0.44) ATMRAB9ACTSSMAPK1GAA
SCHEMBL4180904 0.76 CTSK (0.48) CTDSP1TDP1L3MBTL1RAB9ACTSS
SCHEMBL13854085 0.76 RORC (0.45) ATMKDM4EPKMCTDSP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869026-A1 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2007-12-26 EP claimed
WO-2006105475-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO claimed
EP-1869026-A1 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2007-12-26 EP disclosed
WO-2006105475-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO disclosed