SCHEMBL5486345

SCHEMBL5486345

Clc1nc(-n2cccn2)ncc1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.40
MAPK1 P28482 2/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NOTUM Q6P988 1/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
MPO P05164 2/20 0.36
PDE10A Q9Y233 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPC1 O15118 1/20 0.35
RORC P51449 3/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5598227 0.74 PIN1 (0.40) ADORA2AALDH1A1
SCHEMBL27991818 0.71 ADORA2A (0.55) ADORA2AMAPK1MAPTHTTNPSR1
SCHEMBL6415423 0.71 DHFR (0.49)
SCHEMBL30288591 0.71 NPC1 (0.49) MAPK1MAPTDRD2DRD4DRD3
SCHEMBL2579619 0.70 ALKBH1 (0.43) LMNA
SCHEMBL5473956 0.69 ADORA2A (0.51) ADORA2AMAPK1MAPTHTTNPSR1
SCHEMBL14574878 0.69 ATP4A (0.43) ADORA2AMAPK1MAPTHTTNPSR1
SCHEMBL11865948 0.69 L3MBTL1 (0.42) ADORA2AMAPTHTTL3MBTL1ALDH1A1
SCHEMBL28328153 0.68 NOTUM (0.52) ADORA2AMAPK1MAPTHTTNPSR1
SCHEMBL29448371 0.68 HSP90AB1 (0.59) MAPTNPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070167421-A1 Pyrimidine derivatives and use thereof as agricultural and horticultural fungicides ITO MASHITO 2007-07-19 US disclosed
CN-1942188-A Pyrimidine derivatives and their use as agricultural and horticultural fungicides BAYER CROPSCIENCE AG (DE) 2007-04-04 CN disclosed
EP-1718305-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS AGRICULTURAL AND HORTICULTURAL FUNGICIDES Bayer CropScience AG (DE) 2006-11-08 EP disclosed
WO-2005079798-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS AGRICULTURAL AND HORTICULTURAL FUNGICIDES BAYER CROPSCIENCE AG (DE) 2005-09-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167421-A1 Pyrimidine derivatives and use thereof as agricultural and horticultural fungicides DPYD, DHFR, TYMP ADORA2A 311/4885MAPK1 3295/4885MAPT 2578/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.