SCHEMBL5487413

SCHEMBL5487413

CON1C(=O)CCC(=O)[C@]1(C)C(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)[CH]Cl)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 15/20 0.38
XIAP P98170 2/20 0.34
MLX Q9UH92 1/20 0.34
CMA1 P23946 1/20 0.33
BIRC2 Q13490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2289363 0.90 ELANE (0.42) ELANEXIAPMLXCMA1
SCHEMBL228960 0.89 ELANE (0.38) ELANEXIAPMLXCMA1
SCHEMBL3276266 0.87 ELANE (0.42) ELANEXIAPMLXCMA1
SCHEMBL8662040 0.87 ELANE (0.40) ELANEXIAPMLXCMA1BIRC2
SCHEMBL230923 0.84 ELANE (0.33) ELANECMA1
SCHEMBL535732 0.83 ACE (0.40)
SCHEMBL4410753 0.81 ELANE (0.38) ELANEXIAPMLXCMA1
SCHEMBL387694 0.81 TACR1 (0.40) ELANEXIAPMLXCMA1
SCHEMBL5494650 0.81 ELANE (0.40) ELANEXIAPMLXCMA1
SCHEMBL8661389 0.78 ELANE (0.36) ELANECMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1793006-A2 Nucleic acid ligands and improved methods for producing the same GILEAD SCIENCES, INC. (US) 2007-06-06 EP disclosed
EP-0724647-A4 NUCLEIC ACID LIGANDS AND IMPROVED METHODS FOR PRODUCING THE SAME GILEAD SCIENCES INC (US) 2003-09-17 EP disclosed
US-6083696-A DETECTION OF BLENDED NUCLEIC ACID LIGANDS OF A TARGET COMPOUND; INCUBATION OF BLENDED NUCLEIC ACID MIXTURE WITH THE TARGET, SEPARATING BLENDED NUCLEIC ACIDS WITH INCREASED RECEPTIVITY, AMPLIFYING BLENDED NUCLEIC ACIDS NEXSTAR PHARMACEUTICALS, INC. (US) 2000-07-04 US disclosed
US-5683867-A NUCLEIC ACID LIGANDS, BLENDING, PARTITIONING AND AMPLIFICATION NEXSTAR PHARMACEUTICALS, INC. (US) 1997-11-04 US disclosed
EP-0724647-A1 NUCLEIC ACID LIGANDS AND IMPROVED METHODS FOR PRODUCING THE SAME NeXstar Pharmaceuticals, Inc. (US) 1996-08-07 EP disclosed
US-5472841-A Partitioning the increased affinity nucleic acids from remainder mixture, amplifying the nucleic acids to yield high affinity nucleic acid NEXSTAR PHARMACEUTICALS, INC. (US) 1995-12-05 US disclosed
WO-1995007364-A1 NUCLEIC ACID LIGANDS AND IMPROVED METHODS FOR PRODUCING THE SAME NEXSTAR PHARMACEUTICALS, INC. (US) 1995-03-16 WO disclosed