SCHEMBL5487533

SCHEMBL5487533

NS(=O)(=O)c1ccc(-n2cnnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.49
CA2 P00918 17/20 0.48
CA12 O43570 15/20 0.48
CA9 Q16790 15/20 0.48
CA1 P00915 15/20 0.48
CA5A P35218 4/20 0.46
CA5B Q9Y2D0 4/20 0.46
CA7 P43166 4/20 0.46
CA6 P23280 3/20 0.46
CA4 P22748 2/20 0.46
CA13 Q8N1Q1 2/20 0.46
CA14 Q9ULX7 2/20 0.46
USP2 O75604 1/20 0.46
TSHR P16473 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
AGO2 Q9UKV8 1/20 0.46
SCN2A Q99250 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28054680 0.83 CYP2C9 (0.47) TSHRALDH1A1LMNACYP1A2CYP2C9
SCHEMBL4408673 0.77 CHRNA7 (0.76) CHRNA7CA2CA12CA9CA1
SCHEMBL2771870 0.77 CA2 (0.56) CA2CA12CA9CA1CA5A
SCHEMBL28002115 0.76 CYP1A2 (0.64) CA12CA9TSHRLMNACYP1A2
SCHEMBL202948 0.74 CA2 (0.81) CA2CA12CA9CA1CA5A
SCHEMBL18109146 0.73 LMNA (0.67) CA2CA12CA9CA1CA5A
SCHEMBL7660151 0.72 CYP1A2 (0.38) TDP1ALDH1A1LMNACYP1A2CYP2C9
SCHEMBL7660833 0.72 CYP1A2 (0.50) TSHRTDP1ALDH1A1LMNACYP1A2
SCHEMBL14204073 0.71 PTGS2 (0.43) CA2CA12CA9CA1CA5A
SCHEMBL1352015 0.70 MAPT (0.56) USP2TSHRTDP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183320-B2 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents ELI LILLY AND COMPANY (US) 2007-02-27 US disclosed