Water

Water

SCHEMBL5492464

CC1(C)C(=CC=C2CCC(C=CC3=[N+](CCCCS(=O)(=O)O)c4ccccc4C3(C)C)=C2Cl)N(CCCCS(=O)(=O)O)c2ccccc21.[OH-]

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQ

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.52
FOLR1 P15328 6/20 0.50
HTR1A P08908 1/20 0.49
PRMT1 Q99873 3/20 0.49
CHRM1 P11229 3/20 0.46
CHRM3 P20309 3/20 0.46
HRH2 P25021 3/20 0.46
MLNR O43193 1/20 0.46
NR1I2 O75469 1/20 0.46
PGR P06401 1/20 0.46
ADRB1 P08588 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
DRD2 P14416 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
CNR1 P21554 1/20 0.46
DRD1 P21728 1/20 0.46
TBXA2R P21731 1/20 0.46
SLC6A2 P23975 1/20 0.46
HTR2C P28335 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL30750794 1.00 PTPN1 (0.52) PTPN1FOLR1HTR1APRMT1CHRM1
Water SCHEMBL5492460 1.00 PTPN1 (0.52) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL12891552 0.99 PTPN1 (0.53) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL14364022 0.99 PTPN1 (0.53) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL9101901 0.99 PTPN1 (0.53) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL9101895 0.99 PTPN1 (0.53) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL15026326 0.99 PTPN1 (0.53) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL15026323 0.96 PTPN1 (0.51) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL14666851 0.96 PTPN1 (0.51) PTPN1FOLR1HTR1APRMT1CHRM1
SCHEMBL12364521 0.96 PTPN1 (0.51) PTPN1FOLR1HTR1APRMT1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294370-B2 Polarizing and optical compensating films for visible, ultraviolet and infrared parts of the electromagnetic spectrum KENT STATE UNIVERSITY (US) 2007-11-13 US claimed
US-20200237670-A1 DYE-STABILIZED NANOPARTICLES AND METHODS OF THEIR MANUFACTURE AND THERAPEUTIC USE MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2020-07-30 US disclosed
US-20180021259-A1 DYE-STABILIZED NANOPARTICLES AND METHODS OF THEIR MANUFACTURE AND THERAPEUTIC USE MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2018-01-25 US disclosed
US-8920673-B2 Phosphonium-based ionic liquids and uses LOS ALAMOS NATIONAL SECURITY, LLC (US) 2014-12-30 US disclosed
US-20140065290-A1 COMPOSITIONS AND METHODS OF USE FOR DETECTION AND IMAGING OF PRINTS BY SURFACE-ENHANCED SPECTROSCOPIC TECHNIQUES UT-BATTELLE, LLC (US) 2014-03-06 US disclosed
US-20130030282-A1 SYNTHESIS AND CHARACTERIZATION OF NEAR IR FLUORESCENT MAGNETIC AND NON-MAGNETIC ALBUMIN NANOPARTICLES FOR BIOMEDICAL APPLICATIONS BAR ILAN UNIVERSITY (IL) 2013-01-31 US disclosed
US-20120138789-A1 Phosphonium-Based Ionic Liquids and Uses LOS ALAMOS NATIONAL SECURITY, LLC (US) 2012-06-07 US disclosed
US-7294370-B2 Polarizing and optical compensating films for visible, ultraviolet and infrared parts of the electromagnetic spectrum KENT STATE UNIVERSITY (US) 2007-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200237670-A1 DYE-STABILIZED NANOPARTICLES AND METHODS OF THEIR MANUFACTURE AND THERAPEUTIC USE TP53, SCNN1B, HCCS PTPN1 158/4885FOLR1 1224/4885HTR1A 4082/4885
US-20180021259-A1 DYE-STABILIZED NANOPARTICLES AND METHODS OF THEIR MANUFACTURE AND THERAPEUTIC USE TP53, HCCS, SCNN1B PTPN1 137/4885FOLR1 1189/4885HTR1A 4397/4885
US-20130030282-A1 SYNTHESIS AND CHARACTERIZATION OF NEAR IR FLUORESCENT MAGNETIC AND NON-MAGNETIC ALBUMIN NANOPARTICLES FOR BIOMEDICAL APPLICATIONS ALB, MB, IK PTPN1 1573/4885FOLR1 32/4885HTR1A 4758/4885
US-20120138789-A1 Phosphonium-Based Ionic Liquids and Uses SRMS, PHOSPHO1, TRMT1L PTPN1 3380/4885FOLR1 4234/4885HTR1A 4680/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.