SCHEMBL5496166

SCHEMBL5496166

O=C(O)C(=Cc1ccc(P(=O)=O)cc1)C(F)F

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.33
JUN P05412 1/20 0.33
CYP3A4 P08684 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CAPN1 P07384 1/20 0.33
CAPN2 P17655 1/20 0.33
AKR1C3 P42330 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HTT P42858 1/20 0.31
CISD1 Q9NZ45 1/20 0.31
KDM4E B2RXH2 1/20 0.31
SLC16A3 O15427 1/20 0.31
HPGD P15428 1/20 0.31
SLC16A1 P53985 1/20 0.31
GPR35 Q9HC97 1/20 0.31
EGFR P00533 1/20 0.31
AKR1C1 Q04828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL563697 0.80 AKR1C3 (0.50) TP53CYP3A4CYP1A2CYP2C9AKR1C3
SCHEMBL16266991 0.75 THRB (0.49) CYP3A4CYP1A2AKR1C3ALDH1A1KDM4E
SCHEMBL5488504 0.75 CA2 (0.39) TP53JUNCYP3A4CYP1A2CYP2C9
SCHEMBL4905786 0.64 TRPA1 (0.47) CYP3A4CYP1A2CYP2C9CYP2C19AKR1C3
SCHEMBL4905778 0.64 TRPA1 (0.47) CYP3A4CYP1A2CYP2C9CYP2C19AKR1C3
SCHEMBL4905770 0.64 TRPA1 (0.47) CYP3A4CYP1A2CYP2C9CYP2C19AKR1C3
SCHEMBL14913574 0.62 CYP1A2 (0.55) CYP3A4CYP1A2CYP2C9CYP2C19AKR1C3
SCHEMBL1563519 0.62 AKR1C3 (0.52) TP53CYP3A4CYP1A2CYP2C9AKR1C3
SCHEMBL563363 0.61 AKR1C3 (0.46) TP53CYP3A4CYP1A2CYP2C9AKR1C3
SCHEMBL3226792 0.61 AKR1C3 (0.55) TP53CYP3A4CYP1A2CYP2C9AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070010428-A1 Inhibitors of signal transduction and activator of transcription 3 BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2007-01-11 US disclosed