SCHEMBL5501181

SCHEMBL5501181

C=CCOc1ccc2c(c1)CC(CCc1ccccc1)O2

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.43
BCHE P06276 1/20 0.41
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CYP3A4 P08684 1/20 0.39
MAOA P21397 4/20 0.39
MAOB P27338 4/20 0.39
GPR84 Q9NQS5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727481 0.89 HRH3 (0.42) HRH3ADRA2AADRA2BADRA2CMAOA
SCHEMBL5505186 0.82 HRH3 (0.55) HRH3CYP3A4
SCHEMBL14435045 0.81 ALOX15 (0.44) CYP3A4
SCHEMBL5502112 0.75 DRD2 (0.45) CYP3A4
SCHEMBL27395867 0.75 MAOB (0.49) HRH3MAOAMAOB
SCHEMBL14435037 0.74 CYP3A4 (0.49) HRH3ADRA2AADRA2BADRA2CCYP3A4
SCHEMBL14446493 0.73 CNR2 (0.41) CYP3A4
SCHEMBL5505040 0.72 AKR1B1 (0.37) HRH3CYP3A4
SCHEMBL7293289 0.72 MAOB (0.51) HRH3MAOAMAOB
SCHEMBL7293295 0.72 MAOB (0.51) HRH3MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070202547-A1 Methods For Detecting Substances Which Bind To The Amyloid Precursor Protein Or Beta Amyloid Fragments, And Binding Compounds MERCK & CO., INC. 2007-08-30 US disclosed
US-20070202547-A1 Methods For Detecting Substances Which Bind To The Amyloid Precursor Protein Or Beta Amyloid Fragments, And Binding Compounds MERCK & CO., INC. 2007-08-30 US disclosed
US-20070202547-A1 Methods For Detecting Substances Which Bind To The Amyloid Precursor Protein Or Beta Amyloid Fragments, And Binding Compounds MERCK & CO., INC. 2007-08-30 US disclosed
EP-1743170-A2 METHODS FOR DETECTING SUBSTANCES WHICH BIND TO THE AMYLOID PRECURSOR PROTEIN OR BETA AMYLOID FRAGMENTS, AND BINDING COMPOUNDS Merck & Co., Inc. (US) 2007-01-17 EP disclosed
WO-2005096730-A2 METHODS FOR DETECTING SUBSTANCES WHICH BIND TO THE AMYLOID PRECURSOR PROTEIN OR BETA AMYLOID FRAGMENTS, AND BINDING COMPOUNDS MERCK & CO., INC. (US) 2005-10-20 WO disclosed
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed