SCHEMBL5502143

SCHEMBL5502143

COc1ccc2nc(N3CCNCC3)nc(C(=O)OC(C)(C)C)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.50
SLC2A1 P11166 1/20 0.49
PDE10A Q9Y233 1/20 0.46
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
KMT2A Q03164 4/20 0.44
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 3/20 0.42
POLB P06746 2/20 0.42
UBE2N P61088 2/20 0.42
APAF1 O14727 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
HTR2A P28223 1/20 0.42
GAA P10253 1/20 0.42
MEN1 O00255 2/20 0.42
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502928 0.83 ALDH1A1 (0.53) NCF1KMT2AALDH1A1KDM4EHPGD
SCHEMBL5502137 0.82 NCF1 (0.49) NCF1PDE10AHTR3EHTR3BHTR3A
SCHEMBL4190466 0.70 NCF1 (0.56) NCF1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2708405 0.70 ADRB2 (0.72) NCF1PDE10AHTR3EHTR3BHTR3A
SCHEMBL27993763 0.69 RBP4 (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
Trifluoroacetic Acid SCHEMBL30619102 0.68 NCF1 (0.50) NCF1PDE10AHTR6HTR1AHTR1D
SCHEMBL4144013 0.68 KDM4E (0.41) NCF1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2848141 0.68 NCF1 (0.52) NCF1PDE10AHTR3EHTR3BHTR3A
SCHEMBL31148436 0.67 HTR2C (0.34) ALDH1A1KDM4E
SCHEMBL6636311 0.67 NCF1 (1.00) NCF1PDE10AHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218353-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA UK LTD (GB) 2007-10-17 EP disclosed
EP-1272185-B1 USE OF QUINAZOLINE DERIVATIVES AS ANGIOGENESIS INHIBITORS ASTRAZENECA AB (SE) 2005-07-27 EP disclosed