SCHEMBL5503597

SCHEMBL5503597

Clc1ccccc1OP(Oc1ccccc1Cl)Oc1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
TSHR P16473 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 2/20 0.39
SLC6A4 P31645 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
PKM P14618 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTT P42858 1/20 0.37
CXCL8 P10145 1/20 0.37
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
DPP4 P27487 1/20 0.35
RXRA P19793 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11553081 0.97 LMNA (0.43) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL11677163 0.97 LMNA (0.43) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL19904701 0.89 DPP4 (0.42) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL9621279 0.89 DPP4 (0.42) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL7937629 0.88 LMNA (0.41) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL19904678 0.86 L3MBTL1 (0.42) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL7602939 0.82 LMNA (0.43) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL5503600 0.80 LMNA (0.42) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL1364726 0.80 LMNA (0.42) LMNATSHRSMN1; SMN2HPGDSLC6A4
SCHEMBL9492349 0.80 ALDH1A1 (0.42) LMNATSHRSMN1; SMN2SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005010028-A1 ALPHA-AMINO ACID BENZOTHIAZOLYLTHIO ESTER AS INTERMEDIATES FOR MANUFACTURE OF ACE INHIBITORS AND PROCESS FOR PREPARATION THEREOF LUPIN LIMITED (IN) 2005-02-03 WO claimed
EP-0262061-B1 PROCESS FOR STABILIZING CHLORINATION MIXTURES OF PHENOL AND/OR CHLOROPHENOLS RHONE-POULENC CHIMIE (FR) 1993-02-24 EP claimed
US-4853153-A USING REDUCING AGENT AND CHLORINATED CYCLIC KETONE RHONE-POULENC CHIMIE (FR) 1989-08-01 US claimed
US-3966697-A CATALYST OF COBALT COMPOUND, ORGANOALUMINUM HALIDE, PHOSPHITE, H-ACIDIC COMPOUND CHEMISCHE WERKE HULS AKTIENGESELLSCHAFT (DT) 1976-06-29 US claimed
WO-2024067610-A1 METHOD FOR PREPARING L-GLUFOSINATE BY USING PHOSPHINE REAGENT 摩珈(上海)生物科技有限公司 2024-04-04 WO disclosed
EP-4168487-A1 CURING OF REACTION RESINS, USING UNSATURATED PEROXIDES AS THE INITIATATOR AND ORGANIC PHOSPHITES AS THE ACCELERATOR Röhm GmbH (DE) 2023-04-26 EP disclosed
CN-115916895-A Curing reaction resins using unsaturated peroxides as initiators and organophosphites as accelerators 罗姆化学有限责任公司 2023-04-04 CN disclosed
WO-2021259596-A1 CURING OF REACTION RESINS, USING UNSATURATED PEROXIDES AS THE INITIATATOR AND ORGANIC PHOSPHITES AS THE ACCELERATOR RÖHM GMBH (DE) 2021-12-30 WO disclosed
US-20120220803-A1 Process for Production of Trialkylphosphine CENTRAL GLASS COMPANY, LIMITED (JP) 2012-08-30 US disclosed
EP-1774410-A1 CHARGE CONTROL AGENT, TONER, IMAGE FORMING METHOD, AND IMAGE FORMING APPARATUS Canon Kabushiki Kaisha (JP) 2007-04-18 EP disclosed
EP-1758949-A2 POLYHYDROXYALKANOATE HAVING VINYL GROUP, ESTER GROUP, CARBOXYL GROUP AND SULFONIC ACID GROUP, AND PRODUCTION METHOD THEREOF Canon Kabushiki Kaisha (JP) 2007-03-07 EP disclosed
EP-1758948-A2 POLYHYDROXYALKANOIC ACID HAVING VINYL, ESTER, CARBOXYL OR SULFONIC ACID GROUP AND PRODUCING METHOD THEREFOR Canon Kabushiki Kaisha (JP) 2007-03-07 EP disclosed
EP-0015080-A1 Process for the stabilization of halogenating compound and stabilized halogenating compositions ELI LILLY AND COMPANY (US) 1980-09-03 EP disclosed
EP-0015079-A1 Halogenating compounds and a process for their production ELI LILLY AND COMPANY (US) 1980-09-03 EP disclosed
EP-0014566-A1 Halogenated beta-lactam compounds and process for their preparation ELI LILLY AND COMPANY (US) 1980-08-20 EP disclosed
EP-0014567-A1 Processes for preparation of beta-lactam compounds ELI LILLY AND COMPANY (US) 1980-08-20 EP disclosed
EP-0013461-A1 Process for the preparation of a segmented thermoplastic elastomer AKZO N.V. (NL) 1980-07-23 EP disclosed
US-4211702-A TRIARYLPHOSPHITE-HALOGEN COMPLEX HALOGENATING AGENT ELI LILLY AND COMPANY (US) 1980-07-08 US disclosed
US-4211547-A HERBICIDES MONSANTO COMPANY (US) 1980-07-08 US disclosed
US-3966697-A CATALYST OF COBALT COMPOUND, ORGANOALUMINUM HALIDE, PHOSPHITE, H-ACIDIC COMPOUND CHEMISCHE WERKE HULS AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed