SCHEMBL5505499

SCHEMBL5505499

CN(CCCNC(=O)[C@H](Cc1cc[c]cc1)NS(=O)(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 1/20 0.49
NPY5R Q15761 1/20 0.49
MMP2 P08253 5/20 0.45
MMP9 P14780 4/20 0.45
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
ADAMTS4 O75173 1/20 0.42
MAPK1 P28482 1/20 0.42
CTSL P07711 2/20 0.41
CTSS P25774 2/20 0.41
CTSK P43235 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CTSB P07858 1/20 0.41
F2 P00734 2/20 0.40
TMPRSS6 Q8IU80 2/20 0.40
PTPN1 P18031 2/20 0.40
BMP1 P13497 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5505502 1.00 AVPR1B (0.49) AVPR1BNPY5RMMP2MMP9ALDH1A1
SCHEMBL3735527 0.83 ALDH1A1 (0.46) AVPR1BNPY5RMMP2MMP9ALDH1A1
SCHEMBL3735522 0.83 ALDH1A1 (0.46) AVPR1BNPY5RMMP2MMP9ALDH1A1
SCHEMBL5509174 0.82 ADAMTS4 (0.46) AVPR1BNPY5RMMP2MMP9ALDH1A1
SCHEMBL4866783 0.81 ITGB3 (0.49) NPY5RMMP2MMP9ALDH1A1MAPT
SCHEMBL4866780 0.81 ITGB3 (0.49) NPY5RMMP2MMP9ALDH1A1MAPT
SCHEMBL3735528 0.81 AVPR1B (0.44) AVPR1BNPY5RMMP2MMP9ALDH1A1
SCHEMBL4857259 0.78 NPY5R (0.62) NPY5RMMP2MMP9ALDH1A1MAPT
SCHEMBL4857262 0.78 NPY5R (0.62) NPY5RMMP2MMP9ALDH1A1MAPT
SCHEMBL4864939 0.77 MMP2 (0.49) NPY5RMMP2MMP9ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812012-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Ceptyr, Inc. (US) 2007-08-01 EP disclosed
WO-2006055525-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CEPTYR, INC. (US) 2006-05-26 WO disclosed