SCHEMBL5505729

SCHEMBL5505729

NC(=O)C(C(=O)NCCC1CNc2ccc(F)cc21)C1CCCCC1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 6/20 0.34
IDO1 P14902 1/20 0.34
PIM1 P11309 2/20 0.33
PIM2 Q9P1W9 2/20 0.33
DPP9 Q86TI2 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
PYGL P06737 4/20 0.33
CTSL P07711 1/20 0.32
EPHX1 P07099 1/20 0.32
MC3R P41968 1/20 0.32
HTR1A P08908 1/20 0.32
HTR1D P28221 1/20 0.32
HTR1F P30939 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6688690 1.00 OPRL1 (0.34) OPRL1IDO1PIM1PIM2DPP9
SCHEMBL6696331 0.82 CTSS (0.37) PIM1PIM2NPC1POLBRAB9A
SCHEMBL5497651 0.81 CTSS (0.40) PIM1PIM2NPC1POLBRAB9A
SCHEMBL6685697 0.78 TRPV1 (0.35) IDO1CTSLHTR1AHTR1DHTR1F
SCHEMBL6687531 0.77 TRPV1 (0.34) IDO1PYGL
SCHEMBL6689424 0.77 TRPV1 (0.34) IDO1PYGL
SCHEMBL6693432 0.76 CTSS (0.41) CTSL
SCHEMBL6686987 0.76 CTSL (0.42) NPC1POLBRAB9APYGLCTSL
SCHEMBL6686227 0.75 CTSS (0.40) POLBCTSL
SCHEMBL6689091 0.75 CTSL (0.41) NPC1POLBRAB9ACTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658267-A4 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2007-08-01 EP disclosed
EP-1658267-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2006-05-24 EP disclosed
WO-2005034848-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2005-04-21 WO disclosed