SCHEMBL5497651

SCHEMBL5497651

O=C(NCCC1CNc2ccc(F)cc21)[C@@H](O)CC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.40
CTSL P07711 8/20 0.40
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
METAP2 P50579 2/20 0.35
METAP1 P53582 2/20 0.35
CTSK P43235 2/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GCK P35557 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6696331 0.89 CTSS (0.37) CTSSCTSLRAB9ANPC1METAP2
SCHEMBL6693432 0.84 CTSS (0.41) CTSSCTSLCTSK
SCHEMBL6688690 0.81 OPRL1 (0.34) CTSLRAB9ANPC1PIM1PIM2
SCHEMBL5505729 0.81 OPRL1 (0.34) CTSLRAB9ANPC1PIM1PIM2
SCHEMBL6689460 0.80 MMP3 (0.40) CTSSCTSL
SCHEMBL6690381 0.80 CTSS (0.46) CTSSCTSLCTSK
SCHEMBL6690326 0.80 CTSS (0.45) CTSSCTSLCTSK
SCHEMBL6690633 0.79 USP30 (0.40) CTSSCTSLCTSK
SCHEMBL6690630 0.79 USP30 (0.41) CTSSCTSLCTSK
SCHEMBL6686203 0.78 BMP1 (0.42) CTSSCTSLNPC1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658267-A4 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2007-08-01 EP disclosed
EP-1658267-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2006-05-24 EP disclosed
WO-2005034848-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2005-04-21 WO disclosed