SCHEMBL5506534

SCHEMBL5506534

O=C(c1ccncc1)c1cc(-c2ccccc2)ccc1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
IKBKB O14920 2/20 0.50
CHUK O15111 2/20 0.50
IKBKE Q14164 1/20 0.50
PKMYT1 Q99640 1/20 0.50
HDAC1 Q13547 1/20 0.49
CDC25B P30305 1/20 0.47
ATM Q13315 1/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP2C9 P11712 2/20 0.46
CYP2C8 P10632 1/20 0.46
POLB P06746 1/20 0.45
STAT3 P40763 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPK14 Q16539 1/20 0.44
GSTA1 P08263 1/20 0.44
DHFR P00374 1/20 0.44
HNF4A P41235 1/20 0.44
MCL1 Q07820 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5959807 0.89 CYP2C9 (0.58) MEN1KMT2AIKBKBCDC25BATM
SCHEMBL20147808 0.81 MEN1 (0.62) MEN1KMT2ACDC25BATMALDH1A1
SCHEMBL13291398 0.80 ITGB1 (0.50) MEN1KMT2ACDC25BATMALDH1A1
SCHEMBL27982332 0.79 KMT2A (0.50) MEN1KMT2AIKBKBCHUKIKBKE
SCHEMBL1198770 0.77 KMT2A (0.51) MEN1KMT2AIKBKBCHUKIKBKE
SCHEMBL1960214 0.77 GSTA1 (0.43) MEN1KMT2AIKBKBALDH1A1GSTA1
SCHEMBL593979 0.76 ACMSD (0.66) IKBKBCDC25BATMSMN1; SMN2GSTA1
SCHEMBL28431907 0.75 CDC25B (0.51) MEN1KMT2AHDAC1CDC25BATM
Acetic Acid SCHEMBL27418041 0.75 CYP2C9 (0.58) MEN1KMT2ACDC25BATMALDH1A1
SCHEMBL6422025 0.75 ALDH1A1 (0.56) MEN1KMT2ACDC25BATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697394-B1 COMT INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed