SCHEMBL5523796

SCHEMBL5523796

O=C(Cl)c1cc(F)c(F)c(OC(Cl)(Cl)Cl)c1F

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
CES2 O00748 2/20 0.33
CES1 P23141 2/20 0.33
POLB P06746 1/20 0.30
APEX1 P27695 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5526757 0.88 ALDH1A1 (0.36) ALDH1A1ALOX15CES2CES1
SCHEMBL605762 0.78 ALDH1A1 (0.39) ALDH1A1ALOX15CES2CES1
SCHEMBL5528987 0.77 CES2 (0.32) CES2CES1
SCHEMBL7811260 0.75 ALDH1A1 (0.37) ALDH1A1ALOX15CA1CA2CA4
SCHEMBL5522939 0.73 EPHX2 (0.36) CA1CA2CA4CES2CES1
SCHEMBL345016 0.72 ALDH1A1 (0.48) ALDH1A1ALOX15CA1CA2CA4
SCHEMBL7813771 0.71 KEAP1 (0.37) CES2CES1KEAP1NFE2L2
SCHEMBL9566656 0.70 KEAP1 (0.34) KEAP1NFE2L2
SCHEMBL18186528 0.70 HSD17B1 (0.38) ALDH1A1ALOX15CES2CES1
SCHEMBL5458697 0.69 HSD17B1 (0.39) ALDH1A1ALOX15CES2CES1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070213339-A1 Quinolone Carboxylic Acid Derivatives for Treatment of Hyperproliferative Conditions BAYER PHARMACEUTICALS CORPORATION (US) 2007-09-13 US disclosed
US-20070213339-A1 Quinolone Carboxylic Acid Derivatives for Treatment of Hyperproliferative Conditions BAYER PHARMACEUTICALS CORPORATION (US) 2007-09-13 US disclosed
US-20070213339-A1 Quinolone Carboxylic Acid Derivatives for Treatment of Hyperproliferative Conditions BAYER PHARMACEUTICALS CORPORATION (US) 2007-09-13 US disclosed
EP-1732897-A1 QUINOLONE CARBOXYLIC ACID DERIVATIVES FOR TREATMENT OF HYPERPROLIFERATIVE CONDITIONS Bayer Pharmaceuticals Corporation (US) 2006-12-20 EP disclosed
WO-2005097752-A1 QUINOLONE CARBOXYLIC ACID DERIVATIVES FOR TREATMENT OF HYPERPROLIFERATIVE CONDITIONS BAYER PHARMACEUTICALS CORPORATION (US) 2005-10-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213339-A1 Quinolone Carboxylic Acid Derivatives for Treatment of Hyperproliferative Conditions TP53, RB1, HRAS ALDH1A1 272/4885ALOX15 1666/4885CA1 4567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.