Gabazine

Gabazine

SCHEMBL5529434

COc1ccc(-c2ccc(=N)n(CCCC(=O)O)n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 16/20 1.00
GABRB2 P47870 16/20 1.00
GABRP O00591 6/20 1.00
GABRD O14764 6/20 1.00
GABRB1 P18505 6/20 1.00
GABRG2 P18507 6/20 1.00
GABRB3 P28472 6/20 1.00
GABRA5 P31644 6/20 1.00
GABRA3 P34903 6/20 1.00
GABRA2 P47869 6/20 1.00
GABRA4 P48169 6/20 1.00
GABRE P78334 6/20 1.00
GABRA6 Q16445 6/20 1.00
GABRG1 Q8N1C3 6/20 1.00
GABRG3 Q99928 6/20 1.00
GABRQ Q9UN88 6/20 1.00
CYP1A2 P05177 1/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C9 P11712 1/20 1.00
ALOX15 P16050 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gabazine SCHEMBL5473649 0.99 GABRA1 (0.98) GABRA1GABRB2GABRPGABRDGABRB1
Gabazine SCHEMBL16320027 0.98 GABRA1 (0.95) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL28620347 0.93 GABRA1 (0.86) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL26665197 0.85 GABRA1 (1.00) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL28635070 0.83 GABRA1 (0.71) GABRA1GABRB2GABRPGABRDGABRB1
Bromide SCHEMBL17927694 0.82 GABRA1 (1.00) GABRA1GABRB2GABRPGABRDGABRB1
Hydrochloric Acid SCHEMBL16320560 0.81 GABRA1 (0.95) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL28635088 0.81 GABRA1 (0.67) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL2739432 0.80 GABRA1 (0.90) GABRA1GABRB2GABRPGABRDGABRB1
SCHEMBL415236 0.79 GABRA1 (0.65) GABRA1GABRB2GABRPGABRDGABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116913-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS TEXAS A & M UNIV SYS (US) 2026-04-30 US disclosed
US-12509487-B2 Neurosteroid compounds and methods for their preparation and use in treating central nervous system disorders THE TEXAS A&M UNIVERSITY SYSTEM (US) 2025-12-30 US disclosed
WO-2025262072-A2 NEURONAL DRUG SCREENING METHOD AND NEW APPLICATIONS FOR DILAZEP AND PENBUTOLOL MIĘDZYNARODOWY INSTYTUT BIOLOGII MOLEKULARNEJ I KOMÓRKOWEJ (PL) 2025-12-26 WO disclosed
EP-4528274-A2 BIOMARKERS FOR NEUROPATHOLOGICAL CONDITIONS AND METHODS FOR DIAGNOSIS AND MONITORING THE EFFICACY OF TREATMENT Instituto de Medicina Molecular João Lobo Antunes (PT) 2025-03-26 EP disclosed
US-12173313-B2 Assembly of functionally integrated human forebrain spheroids and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-12-24 US disclosed
EP-4125999-B1 TRKB-FL BASED POLYPEPTIDES AND THEIR USE IN THE TREATMENT OF ALZHEIMER'S DISEASE INST DE MEDICINA MOLECULAR JOAO LOBO ANTUNES (PT) 2024-11-06 EP disclosed
US-20240325760-A1 METHODS FOR DETECTING AND PREVENTING ALZHEIMER'S DISEASE AND MILD COGNITIVE IMPAIRMENT RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2024-10-03 US disclosed
EP-4433468-A1 COMPOSITIONS AND METHODS FOR PRESERVING AND/OR RESTORING NEURAL FUNCTION The Regents of the University of California (US) 2024-09-25 EP disclosed
US-20240034765-A1 SCG2 NEUROPEPTIDES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2024-02-01 US disclosed
EP-3600362-B1 ASSEMBLY OF FUNCTIONALLY INTEGRATED HUMAN FOREBRAIN SPHEROIDS AND METHODS OF USE THEREOF UNIV LELAND STANFORD JUNIOR (US) 2023-12-13 EP disclosed
US-20120122874-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR TREATING DEPRESSION Sunovion Inc. (US) 2012-05-17 US disclosed
US-20120122874-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR TREATING DEPRESSION Sunovion Inc. (US) 2012-05-17 US disclosed
US-8097625-B2 Combination of sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression SUNOVION PHARMACEUTICALS INC. (US) 2012-01-17 US disclosed
US-8097625-B2 Combination of sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression SUNOVION PHARMACEUTICALS INC. (US) 2012-01-17 US disclosed
EP-2343073-A2 Combination of a sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression Sepracor Inc. (US) 2011-07-13 EP disclosed
US-20070299055-A1 COMBINATION OF SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION SEPRACOR INC. (US) 2007-12-27 US disclosed
US-20070299055-A1 COMBINATION OF SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION SEPRACOR INC. (US) 2007-12-27 US disclosed
WO-2005063297-A2 MELATONIN COMBINATION THERAPY FOR IMPROVING SLEEP QUALITY SEPRACOR INC. (US) 2005-07-14 WO disclosed
WO-2005063248-A1 MODAFINIL COMBINATION THERAPY FOR IMPROVING SLEEP QUALITY SEPRACOR INC. (US) 2005-07-14 WO disclosed
WO-2005060968-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION SEPRACOR INC. (US) 2005-07-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299055-A1 COMBINATION OF SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION HTR2A, HTR5A, HTR2C GABRA1 54/4885GABRB2 61/4885GABRP 72/4885
US-12509487-B2 Neurosteroid compounds and methods for their preparation and use in treating central nervous system disorders SLC6A11, GABRE, SLC6A13 GABRA1 29/4885GABRB2 33/4885GABRP 27/4885
US-20120122874-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR TREATING DEPRESSION HTR2A, HTR5A, HTR2C GABRA1 46/4885GABRB2 58/4885GABRP 74/4885
US-20260116913-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS CHRNA9, HSD3B2, HSD3B1 GABRA1 279/4885GABRB2 241/4885GABRP 246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.