SCHEMBL5540348

SCHEMBL5540348

COc1cccc(C(=O)NC2N=CC3=CN(C(=O)c4ccnc(Cl)c4)CCC3=N2)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
ABL1 P00519 3/20 0.39
BCR P11274 3/20 0.39
WNK1 Q9H4A3 1/20 0.39
MGLL Q99685 3/20 0.38
GRM5 P41594 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
MCHR1 Q99705 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
PDE2A O00408 1/20 0.36
PDE3A Q14432 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5538116 0.82 SMN1; SMN2 (0.41) ALDH1A1GRM5TSHRMCHR1
SCHEMBL5546584 0.76 MAPK1 (0.46) ALDH1A1HPGDTSHR
SCHEMBL5540358 0.75 KCNQ3 (0.42) ALDH1A1HPGDABL1BCRWNK1
SCHEMBL5540977 0.75 DRD4 (0.46) MGLLMCHR1
SCHEMBL5545011 0.69 NPC1 (0.41) ALDH1A1HPGD
SCHEMBL3528320 0.66 KDR (0.63) ALDH1A1HPGDGRM5KCNQ3KCNQ2
SCHEMBL5544889 0.65 ALDH1A1 (0.46) ALDH1A1L3MBTL1
SCHEMBL16461033 0.61 RAB9A (0.70) ALDH1A1HPGDTSHR
SCHEMBL2468483 0.60 NPC1 (0.71) ALDH1A1HPGDGRM5TSHRMCHR1
SCHEMBL10339477 0.60 TAS1R3 (0.51) ALDH1A1KCNQ3KCNQ2TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed