SCHEMBL5544949

SCHEMBL5544949

O=C(NC1=NCC2=CN(C(=O)c3c(F)cccc3Cl)CCC2=N1)c1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 2/20 0.36
ABL1 P00519 1/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 2/20 0.36
RORC P51449 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CNR2 P34972 1/20 0.35
GRM5 P41594 1/20 0.34
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34
KCNE1 P15382 1/20 0.34
KCNQ1 P51787 1/20 0.34
KCNQ5 Q9NR82 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545053 0.82 GRM5 (0.39) ALDH1A1L3MBTL1RAB9ANPC1MEN1
SCHEMBL5538119 0.76 RAB9A (0.46) ALDH1A1RAB9ASMN1; SMN2NPC1MEN1
SCHEMBL5544945 0.73 GRM5 (0.38) ALDH1A1L3MBTL1GAARAB9ASMN1; SMN2
SCHEMBL5548741 0.73 SMN1; SMN2 (0.41) ALDH1A1RAB9ASMN1; SMN2NPC1MEN1
SCHEMBL5548545 0.72 SIRT2 (0.42) SMN1; SMN2MEN1KMT2A
SCHEMBL5540380 0.72 ALDH1A1 (0.48) ALDH1A1L3MBTL1GAANPC1MEN1
SCHEMBL5546603 0.71 HPGDS (0.39) ALDH1A1L3MBTL1RAB9ASMN1; SMN2NPC1
SCHEMBL5548146 0.70 MAPT (0.48) ALDH1A1GAARAB9ASMN1; SMN2MEN1
SCHEMBL5546854 0.70 CYP2C19 (0.40) ALDH1A1GAARAB9ASMN1; SMN2NPC1
SCHEMBL5545017 0.70 ALDH1A1 (0.41) ALDH1A1RAB9ASMN1; SMN2NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed