SCHEMBL5550145

SCHEMBL5550145

CC1CCCCN1CCCNc1nc(C(C)(C)C)cn2c(=O)[nH]nc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.42
LMNA P02545 1/20 0.40
KDM4E B2RXH2 5/20 0.40
HSD17B10 Q99714 5/20 0.40
CYP3A4 P08684 5/20 0.40
ALDH1A1 P00352 4/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CXCR4 P61073 6/20 0.40
HPGD P15428 3/20 0.39
THRB P10828 1/20 0.39
MAPK1 P28482 1/20 0.39
FGFR1 P11362 1/20 0.36
TP53 P04637 1/20 0.36
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5549838 0.84 PGK1 (0.40)
SCHEMBL5549394 0.81 PGK1 (0.39) FGFR1
SCHEMBL5550007 0.81 KAT2B (0.39) CYP3A4TSHRMEN1KMT2A
SCHEMBL5548887 0.80 KAT2B (0.40) CYP3A4TSHRMEN1KMT2A
SCHEMBL3526664 0.79 GAA (0.45) LMNAKDM4EHSD17B10ALDH1A1TSHR
SCHEMBL5549024 0.79 KAT2B (0.41) LMNA
SCHEMBL5548632 0.78 KDM1A (0.40) MEN1KMT2A
SCHEMBL5545569 0.76 DRD2 (0.41) LMNAKDM4EHSD17B10CYP3A4ALDH1A1
SCHEMBL3521844 0.76 MAT2A (0.38) KDM4EHSD17B10ALDH1A1MAPK1
SCHEMBL5545560 0.76 GSK3A (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed