SCHEMBL5554486

SCHEMBL5554486

O=C(O)NCCCNCCc1cccc(F)c1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.50
CNR1 P21554 1/20 0.49
TP53 P04637 1/20 0.47
NOS1 P29475 2/20 0.47
NOS3 P29474 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
MARS1 P56192 1/20 0.45
MPO P05164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5117230 0.88 CNR1 (0.59) TAAR1CNR1TP53
SCHEMBL5037823 0.81 CTSS (0.48) TAAR1CNR1MEN1KMT2A
SCHEMBL3054084 0.81 FFAR1 (0.55) TAAR1CNR1TP53NOS1NOS3
SCHEMBL12500551 0.80 TAAR1 (0.65) TAAR1TP53NOS1NOS3KDM4E
SCHEMBL27598565 0.79 TAAR1 (0.56) TAAR1CNR1TP53NOS1NOS3
SCHEMBL28761382 0.79 SIGMAR1 (0.68)
SCHEMBL18191582 0.78 MPO (0.54) KDM4EMEN1KMT2AMPO
SCHEMBL16246990 0.77 ALDH1A1 (0.52) KDM4EMARS1
SCHEMBL5503782 0.77 NOS1 (0.50) TAAR1NOS1NOS3KDM4EMPO
SCHEMBL31114405 0.77 TAAR1 (0.67) TAAR1NOS1NOS3KDM4EMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797099-A1 PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS Epix Delaware, Inc. (US) 2007-06-20 EP disclosed
WO-2006034511-A1 PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS EPIX DELAWARE, INC. (US) 2006-03-30 WO disclosed