SCHEMBL5556232

SCHEMBL5556232

CCCCCC1Cc2ccccc2N1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.51
NOTUM Q6P988 1/20 0.46
ALDH1A1 P00352 4/20 0.45
PRKCD Q05655 4/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP3A4 P08684 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPC1 O15118 1/20 0.43
CYP2C19 P33261 1/20 0.43
ACE P12821 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7593171 0.84 NOTUM (0.57) PKMNOTUMALDH1A1CYP1A2CYP2D6
SCHEMBL7993369 0.84 DRD2 (0.54) PKMNOTUMALDH1A1CYP1A2CYP2D6
SCHEMBL30681441 0.79 DRD2 (0.53) NOTUMALDH1A1CYP1A2NPC1CYP2C19
SCHEMBL7554164 0.79 DRD2 (0.53) NOTUMALDH1A1CYP1A2NPC1CYP2C19
SCHEMBL4289075 0.79 DRD2 (0.53) NOTUMALDH1A1CYP1A2NPC1CYP2C19
SCHEMBL30681525 0.77 NOTUM (0.48) NOTUMALDH1A1CYP1A2NPC1CYP2C19
SCHEMBL28240256 0.77 MTNR1A (0.48) PKMACE
SCHEMBL4285459 0.76 NOTUM (0.42) NOTUMALDH1A1CYP1A2NPC1CYP2C19
SCHEMBL14229140 0.76 NOTUM (0.50) PKMNOTUMALDH1A1CYP1A2CYP2D6
SCHEMBL4386325 0.74 NOTUM (0.44) NOTUMALDH1A1CYP1A2NPC1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833789-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY ENRICHED INDOLINE-2-CARBOXYLIC ACID DSMIP Assets B.V. (NL) 2007-09-19 EP disclosed
WO-2006069799-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY ENRICHED INDOLINE-2-CARBOXYLIC ACID DSM IP ASSETS B.V. (NL) 2006-07-06 WO disclosed
US-6121460-A Process for the preparation of an optically active indoline-2-carboxylic acid or derivative thereof DSM N.V. (NL) 2000-09-19 US disclosed