SCHEMBL5559153

SCHEMBL5559153

Cc1c(C(C)C(=O)OC2CCCC2)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
PTGS2 P35354 1/20 0.36
HSD11B1 P28845 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP19A1 P11511 1/20 0.34
HPGD P15428 2/20 0.33
HCRTR1 O43613 1/20 0.32
PGR P06401 1/20 0.32
KMT2A Q03164 1/20 0.32
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
SLC6A3 Q01959 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822558 0.93 PTGS2 (0.34) TSHRPTGS2CYP19A1KCNH2
SCHEMBL5796692 0.91 PTGS2 (0.37) PTGS2HSD11B1ALDH1A1CYP19A1KMT2A
SCHEMBL5801005 0.91 PTGS2 (0.44) PTGS2CYP19A1SMN1; SMN2
SCHEMBL5800554 0.90 PTGS2 (0.38) TSHRPTGS2HSD11B1SIGMAR1CYP1A2
SCHEMBL5801342 0.90 PTGS2 (0.35) PTGS2HSD11B1ALDH1A1CYP19A1KMT2A
SCHEMBL5559471 0.90 PTGS2 (0.42) PTGS2
SCHEMBL5798160 0.89 L3MBTL1 (0.37) PTGS2HSD11B1ALDH1A1CYP19A1SLC6A3
SCHEMBL5800295 0.88 TSHR (0.36) TSHRPTGS2HSD11B1SIGMAR1CYP1A2
SCHEMBL5797664 0.88 LMNA (0.38) PTGS2HSD11B1CYP3A4ALDH1A1CYP19A1
SCHEMBL5800837 0.87 L3MBTL1 (0.37) PTGS2HSD11B1ALDH1A1SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed