SCHEMBL5800516

SCHEMBL5800516

CC(=O)Oc1c(C)n(C(=O)c2ccc(Cl)c(Cl)c2)c2ccc(O)c(F)c12

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.35
HPGD P15428 1/20 0.34
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
PTGS2 P35354 4/20 0.34
TSHR P16473 1/20 0.34
SLC22A12 Q96S37 1/20 0.33
PTGS1 P23219 2/20 0.33
HSD11B1 P28845 1/20 0.33
PKM P14618 1/20 0.33
CXCL12 P48061 1/20 0.32
F2 P00734 1/20 0.32
PLAU P00749 1/20 0.32
KLKB1 P03952 1/20 0.32
ELANE P08246 1/20 0.32
NOTUM Q6P988 1/20 0.32
SRD5A2 P31213 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800435 0.93 MAOB (0.35) ABCB11AKR1C3AKR1C2PTGS2SLC22A12
SCHEMBL5799149 0.88 AKR1C3 (0.43) ABCB11AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5561193 0.87 HPGD (0.34) HPGDAKR1C3AKR1C2PTGS2TSHR
SCHEMBL5814619 0.86 CNR1 (0.38) ABCB11AKR1C3AKR1C2PTGS2HSD11B1
SCHEMBL5559110 0.81 MAOB (0.35) AKR1C3AKR1C2PTGS2SLC22A12PTGS1
SCHEMBL5560264 0.81 PTGS2 (0.35) ABCB11HPGDAKR1C3AKR1C2PTGS2
SCHEMBL5554202 0.81 TACR3 (0.33) AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5554445 0.80 PPARG (0.37) AKR1C3AKR1C2HSD11B1
SCHEMBL6025591 0.79 PTGS2 (0.48) ABCB11HPGDAKR1C3AKR1C2PTGS2
SCHEMBL5556113 0.79 AKR1C3 (0.53) ABCB11AKR1C3AKR1C2PTGS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed