SCHEMBL5559110

SCHEMBL5559110

CC(=O)Oc1c(C)n(C(=O)c2ccc(Cl)c(F)c2)c2ccc(O)c(C(C)(C)C)c12

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.35
AKR1C3 P42330 2/20 0.32
AKR1C2 P52895 2/20 0.32
PTGS2 P35354 2/20 0.32
TACR3 P29371 5/20 0.31
TACR2 P21452 4/20 0.31
TACR1 P25103 3/20 0.31
SLC22A12 Q96S37 1/20 0.31
RORC P51449 1/20 0.31
PTGS1 P23219 2/20 0.31
KCNH2 Q12809 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
KCNE1 P15382 1/20 0.30
KCNQ1 P51787 1/20 0.30
KCNQ5 Q9NR82 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800435 0.88 MAOB (0.35) MAOBAKR1C3AKR1C2PTGS2TACR3
SCHEMBL5560487 0.81 PDE2A (0.37) MAOBAKR1C3AKR1C2PTGS2TACR3
SCHEMBL5560527 0.81 PTGS2 (0.33) MAOBAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5800516 0.81 ABCB11 (0.35) AKR1C3AKR1C2PTGS2SLC22A12PTGS1
SCHEMBL5554202 0.81 TACR3 (0.33) MAOBAKR1C3AKR1C2PTGS2TACR3
SCHEMBL5560927 0.80 GAA (0.35) AKR1C3AKR1C2
SCHEMBL5559667 0.79 PTGS2 (0.35) MAOBAKR1C3AKR1C2PTGS2TACR3
SCHEMBL5800412 0.79 PTGS2 (0.46) MAOBAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5553743 0.75 AKR1C3 (0.35) MAOBAKR1C3AKR1C2PTGS2SLC22A12
SCHEMBL6464344 0.75 AKR1C3 (0.35) MAOBAKR1C3AKR1C2PTGS2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed