SCHEMBL5559667

SCHEMBL5559667

CC(=O)Oc1c(C)n(C(=O)c2ccc(Cl)c(F)c2)c2cc(F)c(O)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.35
PTGS1 P23219 3/20 0.35
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
SLC22A12 Q96S37 1/20 0.33
ABCB1 P08183 1/20 0.33
MAOB P27338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RORC P51449 1/20 0.33
ABCB11 O95342 1/20 0.33
KDR P35968 1/20 0.32
PREP P48147 1/20 0.32
CELA1 Q9UNI1 1/20 0.32
SRC P12931 1/20 0.32
PDE2A O00408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560264 0.94 PTGS2 (0.35) PTGS2PTGS1AKR1C3AKR1C2SLC22A12
SCHEMBL5800049 0.90 KMT2A (0.37) PTGS2PTGS1AKR1C3AKR1C2SLC22A12
SCHEMBL5800412 0.87 PTGS2 (0.46) PTGS2PTGS1AKR1C3AKR1C2ABCB1
SCHEMBL5553811 0.87 MAPT (0.40) PTGS2AKR1C3AKR1C2KDM4ETP53
SCHEMBL5560588 0.86 MAPT (0.39) PTGS2AKR1C3AKR1C2KDM4ETP53
SCHEMBL5559414 0.85 LMNA (0.40) AKR1C3AKR1C2KDM4ETP53GAA
SCHEMBL5558604 0.83 SRC (0.47) AKR1C3AKR1C2KDM4EHSD17B10SRC
SCHEMBL5554202 0.83 TACR3 (0.33) PTGS2PTGS1AKR1C3AKR1C2MAOB
SCHEMBL5800435 0.82 MAOB (0.35) PTGS2PTGS1AKR1C3AKR1C2SLC22A12
SCHEMBL5558979 0.81 AKR1C3 (0.39) AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed